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Development of new TAK-285 derivatives as potent EGFR/HER2 inhibitors possessing antiproliferative effects against 22RV1 and PC3 prostate carcinoma cell lines.
Son, Seohyun; Elkamhawy, Ahmed; Gul, Anam Rana; Al-Karmalawy, Ahmed A; Alnajjar, Radwan; Abdeen, Ahmed; Ibrahim, Samah F; Alshammari, Saud O; Alshammari, Qamar A; Choi, Won Jun; Park, Tae Jung; Lee, Kyeong.
Afiliación
  • Son S; College of Pharmacy, BK21 FOUR Team and Integrated Research Institute for Drug Development, Dongguk University-Seoul, Goyang, Republic of Korea.
  • Elkamhawy A; College of Pharmacy, BK21 FOUR Team and Integrated Research Institute for Drug Development, Dongguk University-Seoul, Goyang, Republic of Korea.
  • Gul AR; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt.
  • Al-Karmalawy AA; Department of Chemistry, Research Institute of Chem-Bio Diagnostic Technology, Chung-Ang University, Seoul, Republic of Korea.
  • Alnajjar R; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Ahram Canadian University, Giza, Egypt.
  • Abdeen A; Department of Chemistry, Faculty of Science, University of Benghazi, Benghazi, Libya.
  • Ibrahim SF; Faculty of Pharmacy, Libyan International Medical University, Benghazi, Libya.
  • Alshammari SO; Department of Chemistry, University of Cape Town, Rondebosch, South Africa.
  • Alshammari QA; Department of Forensic Medicine and Toxicology, Faculty of Veterinary Medicine, Benha University, Toukh, Egypt.
  • Choi WJ; Department of Clinical Sciences, College of Medicine, Princess Nourah bint Abdulrahman University, Riyadh, Saudi Arabia.
  • Park TJ; Department of Plant Chemistry and Natural Products, Faculty of Pharmacy, Northern Border University, Arar, Saudi Arabia.
  • Lee K; Department of Pharmacology and Toxicology, Faculty of Pharmacy, Northern Border University, Arar, Saudi Arabia.
J Enzyme Inhib Med Chem ; 38(1): 2202358, 2023 Dec.
Article en En | MEDLINE | ID: mdl-37096560

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Neoplasias de la Próstata / Carcinoma / Antineoplásicos Límite: Humans / Male Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Neoplasias de la Próstata / Carcinoma / Antineoplásicos Límite: Humans / Male Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article