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2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms.
Sequeira, Lisa; Distinto, Simona; Meleddu, Rita; Gaspari, Marco; Angeli, Andrea; Cottiglia, Filippo; Secci, Daniela; Onali, Alessia; Sanna, Erica; Borges, Fernanda; Uriarte, Eugenio; Alcaro, Stefano; Supuran, Claudiu T; Maccioni, Elias.
Afiliación
  • Sequeira L; Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria, Monserrato, Italy.
  • Distinto S; CIQUP-IMS/Department of Chemistry and Biochemistry, Faculty of Sciences, University of Porto, Porto, Portugal.
  • Meleddu R; Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria, Monserrato, Italy.
  • Gaspari M; Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria, Monserrato, Italy.
  • Angeli A; Department of Experimental and Clinical Medicine, Research Centre for Advanced Biochemistry and Molecular Biology, "Magna Græcia" University of Catanzaro, Catanzaro, Italy.
  • Cottiglia F; Department of NEUROFARBA, Section of Pharmaceutical Sciences, University of Florence, Florence, Italy.
  • Secci D; Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria, Monserrato, Italy.
  • Onali A; Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria, Monserrato, Italy.
  • Sanna E; Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria, Monserrato, Italy.
  • Borges F; Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria, Monserrato, Italy.
  • Uriarte E; CIQUP-IMS/Department of Chemistry and Biochemistry, Faculty of Sciences, University of Porto, Porto, Portugal.
  • Alcaro S; Department of Organic Chemistry, Faculty of Pharmacy, University of Santiago de Compostela, Santiago de Compostela, Spain.
  • Supuran CT; Department of Health Sciences, "Magna Græcia" University of Catanzaro, Catanzaro, Italy.
  • Maccioni E; Department of NEUROFARBA, Section of Pharmaceutical Sciences, University of Florence, Florence, Italy.
J Enzyme Inhib Med Chem ; 38(1): 2270183, 2023 Dec.
Article en En | MEDLINE | ID: mdl-37870190

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Anhidrasas Carbónicas / Neoplasias Límite: Humans Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Italia

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Anhidrasas Carbónicas / Neoplasias Límite: Humans Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Italia