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Structure-based design of SARS-CoV-2 papain-like protease inhibitors.
Jadhav, Prakash; Huang, Bo; Osipiuk, Jerzy; Zhang, Xiaoming; Tan, Haozhou; Tesar, Christine; Endres, Michael; Jedrzejczak, Robert; Tan, Bin; Deng, Xufang; Joachimiak, Andrzej; Cai, Jianfeng; Wang, Jun.
Afiliación
  • Jadhav P; Department of Medicinal Chemistry, Ernest Mario School of Pharmacy, Rutgers, The State University of New Jersey, Piscataway, NJ, 08854, USA.
  • Huang B; Department of Chemistry, University of South Florida, Tampa, FL, 33620, USA.
  • Osipiuk J; Structural Biology Center, X-ray Science Division, Argonne National Laboratory, Lemont, IL, 60439, USA.
  • Zhang X; Department Physiological Sciences, College of Veterinary Medicine, Oklahoma State University, Stillwater, OK, 74078, USA.
  • Tan H; Department of Medicinal Chemistry, Ernest Mario School of Pharmacy, Rutgers, The State University of New Jersey, Piscataway, NJ, 08854, USA.
  • Tesar C; Structural Biology Center, X-ray Science Division, Argonne National Laboratory, Lemont, IL, 60439, USA; Center for Structural Biology of Infectious Diseases, Consortium for Advanced Science and Engineering, University of Chicago, Chicago, IL, 60667, USA.
  • Endres M; Structural Biology Center, X-ray Science Division, Argonne National Laboratory, Lemont, IL, 60439, USA; Center for Structural Biology of Infectious Diseases, Consortium for Advanced Science and Engineering, University of Chicago, Chicago, IL, 60667, USA.
  • Jedrzejczak R; Structural Biology Center, X-ray Science Division, Argonne National Laboratory, Lemont, IL, 60439, USA; Center for Structural Biology of Infectious Diseases, Consortium for Advanced Science and Engineering, University of Chicago, Chicago, IL, 60667, USA.
  • Tan B; Department of Medicinal Chemistry, Ernest Mario School of Pharmacy, Rutgers, The State University of New Jersey, Piscataway, NJ, 08854, USA.
  • Deng X; Department Physiological Sciences, College of Veterinary Medicine, Oklahoma State University, Stillwater, OK, 74078, USA; Oklahoma Center for Respiratory and Infectious Diseases, Oklahoma State University, Stillwater, OK, 74078, USA.
  • Joachimiak A; Structural Biology Center, X-ray Science Division, Argonne National Laboratory, Lemont, IL, 60439, USA; Center for Structural Biology of Infectious Diseases, Consortium for Advanced Science and Engineering, University of Chicago, Chicago, IL, 60667, USA; Department of Biochemistry and Molecular Biol
  • Cai J; Department of Chemistry, University of South Florida, Tampa, FL, 33620, USA. Electronic address: jianfengcai@usf.edu.
  • Wang J; Department of Medicinal Chemistry, Ernest Mario School of Pharmacy, Rutgers, The State University of New Jersey, Piscataway, NJ, 08854, USA. Electronic address: junwang@pharmacy.rutgers.edu.
Eur J Med Chem ; 264: 116011, 2024 Jan 15.
Article en En | MEDLINE | ID: mdl-38065031

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Papaína / COVID-19 Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2024 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Papaína / COVID-19 Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2024 Tipo del documento: Article País de afiliación: Estados Unidos