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Discovery of AM-1638: A Potent and Orally Bioavailable GPR40/FFA1 Full Agonist.
Brown, Sean P; Dransfield, Paul J; Vimolratana, Marc; Jiao, XianYun; Zhu, Liusheng; Pattaropong, Vatee; Sun, Ying; Liu, Jinqian; Luo, Jian; Zhang, Jane; Wong, Simon; Zhuang, Run; Guo, Qi; Li, Frank; Medina, Julio C; Swaminath, Gayathri; Lin, Daniel C-H; Houze, Jonathan B.
Afiliação
  • Brown SP; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Dransfield PJ; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Vimolratana M; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Jiao X; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Zhu L; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Pattaropong V; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Sun Y; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Liu J; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Luo J; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Zhang J; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Wong S; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Zhuang R; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Guo Q; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Li F; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Medina JC; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Swaminath G; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Lin DC; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
  • Houze JB; Departments of Therapeutic Discovery, Metabolic Disorders, Pharmaceutics and Pharmacokinetic and Drug Metabolism, Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.
ACS Med Chem Lett ; 3(9): 726-30, 2012 Sep 13.
Article em En | MEDLINE | ID: mdl-24900539

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: ACS Med Chem Lett Ano de publicação: 2012 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: ACS Med Chem Lett Ano de publicação: 2012 Tipo de documento: Article País de afiliação: Estados Unidos