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9H-Carbazole-1-carboxamides as potent and selective JAK2 inhibitors.
Zimmermann, Kurt; Sang, Xiaopeng; Mastalerz, Harold A; Johnson, Walter L; Zhang, Guifen; Liu, Qingjie; Batt, Douglas; Lombardo, Louis J; Vyas, Dinesh; Trainor, George L; Tokarski, John S; Lorenzi, Matthew V; You, Dan; Gottardis, Marco M; Lippy, Jonathan; Khan, Javed; Sack, John S; Purandare, Ashok V.
Afiliação
  • Zimmermann K; Bristol-Myers Squibb Co., 5 Research Parkway, Wallingford, CT 06492-1951, USA. Electronic address: Kurt.Zimmermann@bms.com.
  • Sang X; Bristol-Myers Squibb Co., 5 Research Parkway, Wallingford, CT 06492-1951, USA.
  • Mastalerz HA; Bristol-Myers Squibb Co., 5 Research Parkway, Wallingford, CT 06492-1951, USA.
  • Johnson WL; Bristol-Myers Squibb Co., 5 Research Parkway, Wallingford, CT 06492-1951, USA.
  • Zhang G; Bristol-Myers Squibb Co., 5 Research Parkway, Wallingford, CT 06492-1951, USA.
  • Liu Q; Bristol-Myers Squibb Co., Province Line Rd., Princeton, NJ 08540-4000, USA.
  • Batt D; Bristol-Myers Squibb Co., Province Line Rd., Princeton, NJ 08540-4000, USA.
  • Lombardo LJ; Bristol-Myers Squibb Co., Province Line Rd., Princeton, NJ 08540-4000, USA.
  • Vyas D; Bristol-Myers Squibb Co., 5 Research Parkway, Wallingford, CT 06492-1951, USA.
  • Trainor GL; Bristol-Myers Squibb Co., Province Line Rd., Princeton, NJ 08540-4000, USA.
  • Tokarski JS; Bristol-Myers Squibb Co., Province Line Rd., Princeton, NJ 08540-4000, USA.
  • Lorenzi MV; Bristol-Myers Squibb Co., Province Line Rd., Princeton, NJ 08540-4000, USA.
  • You D; Bristol-Myers Squibb Co., Province Line Rd., Princeton, NJ 08540-4000, USA.
  • Gottardis MM; Bristol-Myers Squibb Co., Province Line Rd., Princeton, NJ 08540-4000, USA.
  • Lippy J; Bristol-Myers Squibb Co., Province Line Rd., Princeton, NJ 08540-4000, USA.
  • Khan J; Bristol-Myers Squibb Co., Province Line Rd., Princeton, NJ 08540-4000, USA.
  • Sack JS; Bristol-Myers Squibb Co., Province Line Rd., Princeton, NJ 08540-4000, USA.
  • Purandare AV; Bristol-Myers Squibb Co., Province Line Rd., Princeton, NJ 08540-4000, USA.
Bioorg Med Chem Lett ; 25(14): 2809-12, 2015 Jul 15.
Article em En | MEDLINE | ID: mdl-25987372

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Inibidores de Proteínas Quinases / Janus Quinase 2 / Amidas Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2015 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Inibidores de Proteínas Quinases / Janus Quinase 2 / Amidas Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2015 Tipo de documento: Article