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Discovery of pyrazolopyrimidine derivatives as novel inhibitors of ataxia telangiectasia and rad3 related protein (ATR).
Ramachandran, Sreekanth A; Jadhavar, Pradeep S; Singh, Manvendra P; Sharma, Ankesh; Bagle, Gaurav N; Quinn, Kevin P; Wong, Po-Yin; Protter, Andrew A; Rai, Roopa; Pham, Son M; Lindquist, Jeffrey N.
Afiliação
  • Ramachandran SA; Integral BioSciences, Pvt. Ltd., C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh, 201306, India.
  • Jadhavar PS; Integral BioSciences, Pvt. Ltd., C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh, 201306, India.
  • Singh MP; Integral BioSciences, Pvt. Ltd., C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh, 201306, India.
  • Sharma A; Integral BioSciences, Pvt. Ltd., C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh, 201306, India.
  • Bagle GN; Integral BioSciences, Pvt. Ltd., C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh, 201306, India.
  • Quinn KP; Medivation, Now Pfizer Inc., 525 Market Street, 36th Floor, San Francisco, CA 94105, United States.
  • Wong PY; Medivation, Now Pfizer Inc., 525 Market Street, 36th Floor, San Francisco, CA 94105, United States.
  • Protter AA; Medivation, Now Pfizer Inc., 525 Market Street, 36th Floor, San Francisco, CA 94105, United States; Current address: Palo Alto Pharmaceutical Consulting Service, United States.
  • Rai R; Medivation, Now Pfizer Inc., 525 Market Street, 36th Floor, San Francisco, CA 94105, United States.
  • Pham SM; Medivation, Now Pfizer Inc., 525 Market Street, 36th Floor, San Francisco, CA 94105, United States.
  • Lindquist JN; Medivation, Now Pfizer Inc., 525 Market Street, 36th Floor, San Francisco, CA 94105, United States. Electronic address: pham.sm@gmail.com.
Bioorg Med Chem Lett ; 27(4): 750-754, 2017 02 15.
Article em En | MEDLINE | ID: mdl-28131712

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirazóis / Piridinas / Pirimidinas / Inibidores de Proteínas Quinases / Proteínas Mutadas de Ataxia Telangiectasia Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Índia

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirazóis / Piridinas / Pirimidinas / Inibidores de Proteínas Quinases / Proteínas Mutadas de Ataxia Telangiectasia Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Índia