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Identification of compound D2923 as a novel anti-tumor agent targeting CSF1R.
Liu, Ying-Qiang; Wang, Ya-Nan; Lu, Xiao-Yun; Tong, Lin-Jiang; Li, Yan; Zhang, Tao; Xun, Qiu-Ju; Feng, Fang; Chen, Yu-Zhe; Su, Yi; Shen, Yan-Yan; Chen, Yi; Geng, Mei-Yu; Ding, Ke; Li, Yan-Li; Xie, Hua; Ding, Jian.
Afiliação
  • Liu YQ; School of Life Science, Shanghai University, 200444, Shanghai, China.
  • Wang YN; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 201203, Shanghai, China.
  • Lu XY; School of Pharmacy, University of Chinese Academy of Sciences, 100049, Beijing, China.
  • Tong LJ; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 201203, Shanghai, China.
  • Li Y; School of Pharmacy, University of Chinese Academy of Sciences, 100049, Beijing, China.
  • Zhang T; School of Life Science and Technology, ShanghaiTech University, 201210, Shanghai, China.
  • Xun QJ; School of Pharmacy, Jinan University, No. 601 Huangpu Avenue, 510632, West Guangzhou, China.
  • Feng F; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 201203, Shanghai, China.
  • Chen YZ; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 201203, Shanghai, China.
  • Su Y; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 201203, Shanghai, China.
  • Shen YY; School of Pharmacy, University of Chinese Academy of Sciences, 100049, Beijing, China.
  • Chen Y; School of Life Science and Technology, ShanghaiTech University, 201210, Shanghai, China.
  • Geng MY; School of Pharmacy, University of Chinese Academy of Sciences, 100049, Beijing, China.
  • Ding K; School of Pharmacy, Jinan University, No. 601 Huangpu Avenue, 510632, West Guangzhou, China.
  • Li YL; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 201203, Shanghai, China.
  • Xie H; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 201203, Shanghai, China.
  • Ding J; School of Pharmacy, University of Chinese Academy of Sciences, 100049, Beijing, China.
Acta Pharmacol Sin ; 39(11): 1768-1776, 2018 Nov.
Article em En | MEDLINE | ID: mdl-29968849

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirimidinonas / Leucemia Mieloide / Receptores de Fator Estimulador das Colônias de Granulócitos e Macrófagos / Inibidores de Proteínas Quinases / Antineoplásicos Tipo de estudo: Diagnostic_studies / Prognostic_studies Limite: Animals / Humans / Male Idioma: En Revista: Acta Pharmacol Sin Assunto da revista: FARMACOLOGIA Ano de publicação: 2018 Tipo de documento: Article País de afiliação: China

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirimidinonas / Leucemia Mieloide / Receptores de Fator Estimulador das Colônias de Granulócitos e Macrófagos / Inibidores de Proteínas Quinases / Antineoplásicos Tipo de estudo: Diagnostic_studies / Prognostic_studies Limite: Animals / Humans / Male Idioma: En Revista: Acta Pharmacol Sin Assunto da revista: FARMACOLOGIA Ano de publicação: 2018 Tipo de documento: Article País de afiliação: China