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Synthesis and Pharmacological Evaluation of 3-[(4-Oxo-4H-pyrido[3,2-e][1,3]thiazin-2-yl)(phenyl)amino]propanenitrile Derivatives as Orally Active AMPA Receptor Antagonists.
Inami, Hiroshi; Shishikura, Jun-Ichi; Yasunaga, Tomoyuki; Hirano, Masaaki; Kimura, Takenori; Yamashita, Hiroshi; Ohno, Kazushige; Sakamoto, Shuichi.
Afiliação
  • Inami H; Drug Discovery Research, Astellas Pharma Inc.
  • Shishikura JI; Drug Discovery Research, Astellas Pharma Inc.
  • Yasunaga T; Drug Discovery Research, Astellas Pharma Inc.
  • Hirano M; Drug Discovery Research, Astellas Pharma Inc.
  • Kimura T; Drug Discovery Research, Astellas Pharma Inc.
  • Yamashita H; Drug Discovery Research, Astellas Pharma Inc.
  • Ohno K; Drug Discovery Research, Astellas Pharma Inc.
  • Sakamoto S; Drug Discovery Research, Astellas Pharma Inc.
Chem Pharm Bull (Tokyo) ; 67(7): 699-706, 2019.
Article em En | MEDLINE | ID: mdl-31257325

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptores de AMPA / Anticonvulsivantes / Nitrilas Limite: Animals Idioma: En Revista: Chem Pharm Bull (Tokyo) Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptores de AMPA / Anticonvulsivantes / Nitrilas Limite: Animals Idioma: En Revista: Chem Pharm Bull (Tokyo) Ano de publicação: 2019 Tipo de documento: Article