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Discovery of HWL-088: A highly potent FFA1/GPR40 agonist bearing a phenoxyacetic acid scaffold.
Li, Zheng; Ren, Qiang; Wang, Xuekun; Zhou, Zongtao; Hu, Lijun; Deng, Liming; Guan, Li; Qiu, Qianqian.
Afiliação
  • Li Z; School of Pharmacy, Guangdong Pharmaceutical University, Guangzhou 510006, PR China.
  • Ren Q; School of Pharmacy, Guangdong Pharmaceutical University, Guangzhou 510006, PR China.
  • Wang X; College of Pharmacy, Liaocheng University, Liaocheng 252059, PR China.
  • Zhou Z; School of Pharmacy, Guangdong Pharmaceutical University, Guangzhou 510006, PR China.
  • Hu L; School of Pharmacy, Guangdong Pharmaceutical University, Guangzhou 510006, PR China.
  • Deng L; School of Pharmacy, Guangdong Pharmaceutical University, Guangzhou 510006, PR China.
  • Guan L; School of Pharmacy, Guangdong Pharmaceutical University, Guangzhou 510006, PR China. Electronic address: guanli@gdpu.edu.cn.
  • Qiu Q; School of Pharmacy, Jiangsu Provincial Key Laboratory of Coastal Wetland Bioresources and Environmental Protection, Yancheng Teachers' University, Yancheng, PR China. Electronic address: qianqianqiu_cpu@126.com.
Bioorg Chem ; 92: 103209, 2019 11.
Article em En | MEDLINE | ID: mdl-31487621

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptores Acoplados a Proteínas G / Diabetes Mellitus Experimental / Diabetes Mellitus Tipo 2 / Descoberta de Drogas / Hipoglicemiantes / Acetatos Tipo de estudo: Prognostic_studies Limite: Animals Idioma: En Revista: Bioorg Chem Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptores Acoplados a Proteínas G / Diabetes Mellitus Experimental / Diabetes Mellitus Tipo 2 / Descoberta de Drogas / Hipoglicemiantes / Acetatos Tipo de estudo: Prognostic_studies Limite: Animals Idioma: En Revista: Bioorg Chem Ano de publicação: 2019 Tipo de documento: Article