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Identification of cysteinyl-leukotriene-receptor 1 antagonists as ligands for the bile acid receptor GPBAR1.
Biagioli, Michele; Carino, Adriana; Marchianò, Silvia; Roselli, Rosalinda; Di Giorgio, Cristina; Bordoni, Martina; Fiorucci, Chiara; Sepe, Valentina; Conflitti, Paolo; Limongelli, Vittorio; Distrutti, Eleonora; Baldoni, Monia; Zampella, Angela; Fiorucci, Stefano.
Afiliação
  • Biagioli M; Department of Surgical and Biomedical Sciences, University of Perugia, via L. Severi 1, 06132 Perugia, Italy. Electronic address: michele.biagioli@live.it.
  • Carino A; Department of Surgical and Biomedical Sciences, University of Perugia, via L. Severi 1, 06132 Perugia, Italy. Electronic address: adriana.carino@unipg.it.
  • Marchianò S; Department of Surgical and Biomedical Sciences, University of Perugia, via L. Severi 1, 06132 Perugia, Italy. Electronic address: silvia4as@hotmail.it.
  • Roselli R; Department of Pharmacy, University of Naples "Federico II", via D. Montesano 49, 80131 Naples, Italy. Electronic address: rosellirosalinda@yahoo.it.
  • Di Giorgio C; Department of Surgical and Biomedical Sciences, University of Perugia, via L. Severi 1, 06132 Perugia, Italy. Electronic address: cristi.digiorgio@gmail.com.
  • Bordoni M; Department of Surgical and Biomedical Sciences, University of Perugia, via L. Severi 1, 06132 Perugia, Italy. Electronic address: mbordoni92@gmail.com.
  • Fiorucci C; Department of Surgical and Biomedical Sciences, University of Perugia, via L. Severi 1, 06132 Perugia, Italy. Electronic address: chiara.fiorucci125@gmail.com.
  • Sepe V; Department of Pharmacy, University of Naples "Federico II", via D. Montesano 49, 80131 Naples, Italy. Electronic address: valentina.sepe@unina.it.
  • Conflitti P; Università della Svizzera Italiana (USI), Faculty of Biomedical Sciences, Institute of Computational Science, Via G. Buffi 13, CH-6900 Lugano, Switzerland. Electronic address: paolo.conflitti@usi.ch.
  • Limongelli V; Department of Pharmacy, University of Naples "Federico II", via D. Montesano 49, 80131 Naples, Italy; Università della Svizzera Italiana (USI), Faculty of Biomedical Sciences, Institute of Computational Science, Via G. Buffi 13, CH-6900 Lugano, Switzerland. Electronic address: vittorio.limongelli@us
  • Distrutti E; SC of Gastroenterology and Hepatology, Azienda Ospedaliera di Perugia, Perugia, Italy. Electronic address: eleonoradistrutti@katamail.com.
  • Baldoni M; Department of Medicine, University of Perugia, via L. Severi 1, 06132 Perugia, Italy. Electronic address: monia.baldoni@unipg.it.
  • Zampella A; Department of Pharmacy, University of Naples "Federico II", via D. Montesano 49, 80131 Naples, Italy. Electronic address: angela.zampella@unina.it.
  • Fiorucci S; Department of Surgical and Biomedical Sciences, University of Perugia, via L. Severi 1, 06132 Perugia, Italy. Electronic address: stefano.fiorucci@unipg.it.
Biochem Pharmacol ; 177: 113987, 2020 07.
Article em En | MEDLINE | ID: mdl-32330496

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinolinas / Anti-Inflamatórios não Esteroides / Receptores de Leucotrienos / Colite / Antagonistas de Leucotrienos / Receptores Acoplados a Proteínas G Tipo de estudo: Diagnostic_studies Limite: Animals / Humans Idioma: En Revista: Biochem Pharmacol Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinolinas / Anti-Inflamatórios não Esteroides / Receptores de Leucotrienos / Colite / Antagonistas de Leucotrienos / Receptores Acoplados a Proteínas G Tipo de estudo: Diagnostic_studies Limite: Animals / Humans Idioma: En Revista: Biochem Pharmacol Ano de publicação: 2020 Tipo de documento: Article