Combined Peptide and Small-Molecule Approach toward Nonacidic THIQ Inhibitors of the KEAP1/NRF2 Interaction.

Ontoria, Jesus M; Biancofiore, Ilaria; Fezzardi, Paola; Ferrigno, Federica; Torrente, Esther; Colarusso, Stefania; Bianchi, Elisabetta; Andreini, Matteo; Patsilinakos, Alexandros; Kempf, Georg; Augustin, Martin; Steinbacher, Stefan; Summa, Vincenzo; Pacifici, Robert; Muñoz-Sanjuan, Ignacio; Park, Larry; Bresciani, Alberto; Dominguez, Celia; Sherman, Leticia Toledo; Harper, Steven

Ontoria, Jesus M; Biancofiore, Ilaria; Fezzardi, Paola; Ferrigno, Federica; Torrente, Esther; Colarusso, Stefania; Bianchi, Elisabetta; Andreini, Matteo; Patsilinakos, Alexandros; Kempf, Georg; Augustin, Martin; Steinbacher, Stefan; Summa, Vincenzo; Pacifici, Robert; Muñoz-Sanjuan, Ignacio; Park, Larry; Bresciani, Alberto; Dominguez, Celia; Sherman, Leticia Toledo; Harper, Steven.

Afiliação

Ontoria JM; IRBM S.p.A., Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
Biancofiore I; IRBM S.p.A., Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
Fezzardi P; IRBM S.p.A., Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
Ferrigno F; IRBM S.p.A., Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
Torrente E; IRBM S.p.A., Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
Colarusso S; IRBM S.p.A., Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
Bianchi E; IRBM S.p.A., Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
Andreini M; IRBM S.p.A., Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
Patsilinakos A; IRBM S.p.A., Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
Kempf G; Proteros Biostructures GmbH, Bunsenstraße 7 a, 82152 Planegg, Germany.
Augustin M; Proteros Biostructures GmbH, Bunsenstraße 7 a, 82152 Planegg, Germany.
Steinbacher S; Proteros Biostructures GmbH, Bunsenstraße 7 a, 82152 Planegg, Germany.
Summa V; IRBM S.p.A., Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
Pacifici R; CHDI Management/CHDI Foundation, 6080 Center Drive, Los Angeles, California 90045, United States.
Muñoz-Sanjuan I; CHDI Management/CHDI Foundation, 6080 Center Drive, Los Angeles, California 90045, United States.
Park L; CHDI Management/CHDI Foundation, 6080 Center Drive, Los Angeles, California 90045, United States.
Bresciani A; IRBM S.p.A., Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
Dominguez C; CHDI Management/CHDI Foundation, 6080 Center Drive, Los Angeles, California 90045, United States.
Sherman LT; CHDI Management/CHDI Foundation, 6080 Center Drive, Los Angeles, California 90045, United States.
Harper S; IRBM S.p.A., Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.

ACS Med Chem Lett ; 11(5): 740-746, 2020 May 14.

Article em En | MEDLINE | ID: mdl-32435379

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Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: ACS Med Chem Lett Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Itália

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