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A FabG inhibitor targeting an allosteric binding site inhibits several orthologs from Gram-negative ESKAPE pathogens.
Vella, Peter; Rudraraju, Reshma Srilakshmi; Lundbäck, Thomas; Axelsson, Hanna; Almqvist, Helena; Vallin, Michaela; Schneider, Gunter; Schnell, Robert.
Afiliação
  • Vella P; Department of Medical Biochemistry and Biophysics, Karolinska Institutet, S-17 165 Stockholm, Sweden.
  • Rudraraju RS; Department of Medical Biochemistry and Biophysics, Karolinska Institutet, S-17 165 Stockholm, Sweden.
  • Lundbäck T; Chemical Biology Consortium Sweden, Science for Life Laboratory, Department of Medical Biochemistry and Biophysics, Karolinska Institutet, S-171 65 Stockholm, Sweden.
  • Axelsson H; Chemical Biology Consortium Sweden, Science for Life Laboratory, Department of Medical Biochemistry and Biophysics, Karolinska Institutet, S-171 65 Stockholm, Sweden.
  • Almqvist H; Chemical Biology Consortium Sweden, Science for Life Laboratory, Department of Medical Biochemistry and Biophysics, Karolinska Institutet, S-171 65 Stockholm, Sweden.
  • Vallin M; Chemical Biology Consortium Sweden, Science for Life Laboratory, Department of Medical Biochemistry and Biophysics, Karolinska Institutet, S-171 65 Stockholm, Sweden.
  • Schneider G; Department of Medical Biochemistry and Biophysics, Karolinska Institutet, S-17 165 Stockholm, Sweden.
  • Schnell R; Department of Medical Biochemistry and Biophysics, Karolinska Institutet, S-17 165 Stockholm, Sweden. Electronic address: Robert.Schnell@ki.se.
Bioorg Med Chem ; 30: 115898, 2021 01 15.
Article em En | MEDLINE | ID: mdl-33388594

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pseudomonas aeruginosa / Salmonella typhimurium / Acinetobacter baumannii / Oxirredutases do Álcool / Inibidores Enzimáticos Idioma: En Revista: Bioorg Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Suécia

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pseudomonas aeruginosa / Salmonella typhimurium / Acinetobacter baumannii / Oxirredutases do Álcool / Inibidores Enzimáticos Idioma: En Revista: Bioorg Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Suécia