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N-Thio-ß-lactams targeting L,D-transpeptidase-2, with activity against drug-resistant strains of Mycobacterium tuberculosis.
Martelli, Giulia; Pessatti, Tomas Bohn; Steiner, Eva Maria; Cirillo, Martina; Caso, Carolina; Bisognin, Francesco; Landreh, Michael; Monte, Paola Dal; Giacomini, Daria; Schnell, Robert.
Afiliação
  • Martelli G; Department of Chemistry "G. Ciamician", University of Bologna, Via Selmi 2, 40126 Bologna, Italy.
  • Pessatti TB; Department of Medical Biochemistry and Biophysics, Karolinska Institutet, 17 165 Stockholm, Sweden.
  • Steiner EM; Department of Medical Biochemistry and Biophysics, Karolinska Institutet, 17 165 Stockholm, Sweden.
  • Cirillo M; Department of Chemistry "G. Ciamician", University of Bologna, Via Selmi 2, 40126 Bologna, Italy.
  • Caso C; Department of Medical Biochemistry and Biophysics, Karolinska Institutet, 17 165 Stockholm, Sweden.
  • Bisognin F; IRCCS Azienda Ospedaliero-Universitaria di Bologna, Microbiology Unit, Via Massarenti, 9, 40138 Bologna, Italy.
  • Landreh M; Department of Microbiology, Tumor and Cell Biology, Karolinska Institutet, 17 165 Stockholm, Sweden.
  • Monte PD; IRCCS Azienda Ospedaliero-Universitaria di Bologna, Microbiology Unit, Via Massarenti, 9, 40138 Bologna, Italy. Electronic address: paola.dalmonte@unibo.it.
  • Giacomini D; Department of Chemistry "G. Ciamician", University of Bologna, Via Selmi 2, 40126 Bologna, Italy. Electronic address: daria.giacomini@unibo.it.
  • Schnell R; Department of Medical Biochemistry and Biophysics, Karolinska Institutet, 17 165 Stockholm, Sweden. Electronic address: robert.schnell@ki.se.
Cell Chem Biol ; 28(9): 1321-1332.e5, 2021 09 16.
Article em En | MEDLINE | ID: mdl-33826941

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Peptidil Transferases / Farmacorresistência Bacteriana / Beta-Lactamas / Antibacterianos / Mycobacterium tuberculosis Idioma: En Revista: Cell Chem Biol Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Itália

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Peptidil Transferases / Farmacorresistência Bacteriana / Beta-Lactamas / Antibacterianos / Mycobacterium tuberculosis Idioma: En Revista: Cell Chem Biol Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Itália