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3H-Pyrazolo[4,3-f]quinoline-Based Kinase Inhibitors Inhibit the Proliferation of Acute Myeloid Leukemia Cells In Vivo.
Dayal, Neetu; Reznícková, Eva; Hernandez, Delmis E; Perina, Miroslav; Torregrosa-Allen, Sandra; Elzey, Bennett D; Skerlová, Jana; Ajani, Haresh; Djukic, Stefan; Vojácková, Veronika; Lepsík, Martin; Rezácová, Pavlína; Krystof, Vladimír; Jorda, Radek; Sintim, Herman O.
Afiliação
  • Dayal N; Department of Chemistry, Purdue University, West Lafayette, Indiana 47907, United States.
  • Reznícková E; Department of Experimental Biology, Faculty of Science, Palacký University Olomouc, Slechtitelu 27, Olomouc 78371, Czech Republic.
  • Hernandez DE; Department of Chemistry, Purdue University, West Lafayette, Indiana 47907, United States.
  • Perina M; Department of Experimental Biology, Faculty of Science, Palacký University Olomouc, Slechtitelu 27, Olomouc 78371, Czech Republic.
  • Torregrosa-Allen S; Purdue University Center for Cancer Research, Purdue University, West Lafayette, Indiana 47907, United States.
  • Elzey BD; Purdue University Center for Cancer Research, Purdue University, West Lafayette, Indiana 47907, United States.
  • Skerlová J; Department of Comparative Pathobiology, Purdue University, West Lafayette, Indiana 47907, United States.
  • Ajani H; Institute of Organic Chemistry and Biochemistry of the Czech Academy of Sciences, Flemingovo Nám. 2, Prague 16610, Czech Republic.
  • Djukic S; Institute of Molecular Genetics of the Czech Academy of Sciences, Vídenská 1083, Prague 14220, Czech Republic.
  • Vojácková V; Institute of Organic Chemistry and Biochemistry of the Czech Academy of Sciences, Flemingovo Nám. 2, Prague 16610, Czech Republic.
  • Lepsík M; Institute of Organic Chemistry and Biochemistry of the Czech Academy of Sciences, Flemingovo Nám. 2, Prague 16610, Czech Republic.
  • Rezácová P; Department of Experimental Biology, Faculty of Science, Palacký University Olomouc, Slechtitelu 27, Olomouc 78371, Czech Republic.
  • Krystof V; Institute of Organic Chemistry and Biochemistry of the Czech Academy of Sciences, Flemingovo Nám. 2, Prague 16610, Czech Republic.
  • Jorda R; Institute of Organic Chemistry and Biochemistry of the Czech Academy of Sciences, Flemingovo Nám. 2, Prague 16610, Czech Republic.
  • Sintim HO; Institute of Molecular Genetics of the Czech Academy of Sciences, Vídenská 1083, Prague 14220, Czech Republic.
J Med Chem ; 64(15): 10981-10996, 2021 08 12.
Article em En | MEDLINE | ID: mdl-34288692

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Leucemia Mieloide Aguda / Inibidores de Proteínas Quinases / Tirosina Quinase 3 Semelhante a fms / Antineoplásicos Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Leucemia Mieloide Aguda / Inibidores de Proteínas Quinases / Tirosina Quinase 3 Semelhante a fms / Antineoplásicos Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Estados Unidos