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Novel Selective and Low-Toxic Inhibitor of LmCPB2.8ΔCTE (CPB) One Important Cysteine Protease for Leishmania Virulence.
Moreira, Vitor Partite; da Silva Mela, Michele Ferreira; Anjos, Luana Ribeiro Dos; Saraiva, Leonardo Figueiredo; Arenas Velásquez, Angela M; Kalaba, Predrag; Fabisiková, Anna; Clementino, Leandro da Costa; Aufy, Mohammed; Studenik, Christian; Gajic, Natalie; Prado-Roller, Alexander; Magalhães, Alvicler; Zehl, Martin; Figueiredo, Ingrid Delbone; Baviera, Amanda Martins; Cilli, Eduardo Maffud; Graminha, Marcia A S; Lubec, Gert; Gonzalez, Eduardo R Perez.
Afiliação
  • Moreira VP; Fine Organic Chemistry Lab, School of Sciences and Technology, São Paulo State University (UNESP), Presidente Prudente 19060-080, Brazil.
  • da Silva Mela MF; School of Pharmaceutical Sciences, São Paulo State University (UNESP), Araraquara 14800-903, Brazil.
  • Anjos LRD; Fine Organic Chemistry Lab, School of Sciences and Technology, São Paulo State University (UNESP), Presidente Prudente 19060-080, Brazil.
  • Saraiva LF; Laboratory of Luminescence in Materials and Sensors, School of Sciences and Technology, São Paulo State University (UNESP), Presidente Prudente 19060-560, Brazil.
  • Arenas Velásquez AM; School of Pharmaceutical Sciences, São Paulo State University (UNESP), Araraquara 14800-903, Brazil.
  • Kalaba P; Department of Pharmaceutical Sciences, Division of Pharmaceutical Chemistry, Faculty of Life Sciences, University of Vienna, Josef Holaubek Platz 2, UZAII, 1090 Vienna, Austria.
  • Fabisiková A; Mass Spectrometry Centre, Faculty of Chemistry, University of Vienna, Währinger Straße 38, 1090 Vienna, Austria.
  • Clementino LDC; School of Pharmaceutical Sciences, São Paulo State University (UNESP), Araraquara 14800-903, Brazil.
  • Aufy M; Department of Pharmaceutical Sciences, Division of Pharmacology and Toxicology, University of Vienna, Josef Holaubek Platz 2, UZAII (2D 259), 1090 Vienna, Austria.
  • Studenik C; Department of Pharmaceutical Sciences, Division of Pharmacology and Toxicology, University of Vienna, Josef Holaubek Platz 2, UZAII (2D 259), 1090 Vienna, Austria.
  • Gajic N; Centre for X-ray Structure Analysis, Faculty of Chemistry, University of Vienna, Währinger Straße 40-42, 1090 Vienna, Austria.
  • Prado-Roller A; Centre for X-ray Structure Analysis, Faculty of Chemistry, University of Vienna, Währinger Straße 40-42, 1090 Vienna, Austria.
  • Magalhães A; Department of Organic Chemistry, Chemistry School, Federal University of Rio de Janeiro, Rio de Janeiro 21941-598, Brazil.
  • Zehl M; Mass Spectrometry Centre, Faculty of Chemistry, University of Vienna, Währinger Straße 38, 1090 Vienna, Austria.
  • Figueiredo ID; Department of Analytical Chemistry, Faculty of Chemistry, University of Vienna, Währinger Straße 38, 1090 Vienna, Austria.
  • Baviera AM; School of Pharmaceutical Sciences, São Paulo State University (UNESP), Araraquara 14800-903, Brazil.
  • Cilli EM; School of Pharmaceutical Sciences, São Paulo State University (UNESP), Araraquara 14800-903, Brazil.
  • Graminha MAS; Department of Biochemistry and Organic Chemistry, Institute of Chemistry, São Paulo State University (UNESP), Araraquara 14800-060, Brazil.
  • Lubec G; School of Pharmaceutical Sciences, São Paulo State University (UNESP), Araraquara 14800-903, Brazil.
  • Gonzalez ERP; Department of Neuroproteomics, Paracelsus Medical University, 5020 Salzburg, Austria.
Biomolecules ; 12(12)2022 12 19.
Article em En | MEDLINE | ID: mdl-36551331

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Leishmaniose / Leishmania major / Cisteína Proteases Limite: Animals Idioma: En Revista: Biomolecules Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Brasil

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Leishmaniose / Leishmania major / Cisteína Proteases Limite: Animals Idioma: En Revista: Biomolecules Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Brasil