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Platform Reagents Enable Synthesis of Ligand-Directed Covalent Probes: Study of Cannabinoid Receptor 2 in Live Cells.
Kosar, Miroslav; Sykes, David A; Viray, Alexander E G; Vitale, Rosa Maria; Sarott, Roman C; Ganzoni, Rudolf L; Onion, David; Tobias, Janelle M; Leippe, Philipp; Ullmer, Christoph; Zirwes, Elisabeth A; Guba, Wolfgang; Grether, Uwe; Frank, James A; Veprintsev, Dmitry B; Carreira, Erick M.
Afiliação
  • Kosar M; Laboratorium für Organische Chemie, Eidgenössische Technische Hochschule Zürich, Vladimir-Prelog-Weg 3, 8093 Zürich, Switzerland.
  • Sykes DA; Centre of Membrane Proteins and Receptors (COMPARE), University of Birmingham and University of Nottingham, Midlands, Nottingham NG7 2UH, U.K.
  • Viray AEG; Faculty of Medicine & Health Sciences, University of Nottingham, Nottingham NG7 2UH, U.K.
  • Vitale RM; Department of Chemical Physiology & Biochemistry, Oregon Health & Science University, Portland, Oregon 97239-3098, United States.
  • Sarott RC; Institute of Biomolecular Chemistry, National Research Council (ICB-CNR), Via Campi Flegrei 34, 80078 Pozzuoli, Italy.
  • Ganzoni RL; Laboratorium für Organische Chemie, Eidgenössische Technische Hochschule Zürich, Vladimir-Prelog-Weg 3, 8093 Zürich, Switzerland.
  • Onion D; Laboratorium für Organische Chemie, Eidgenössische Technische Hochschule Zürich, Vladimir-Prelog-Weg 3, 8093 Zürich, Switzerland.
  • Tobias JM; School of Life Sciences, University of Nottingham, Nottingham NG7 2UH, U.K.
  • Leippe P; Department of Chemical Physiology & Biochemistry, Oregon Health & Science University, Portland, Oregon 97239-3098, United States.
  • Ullmer C; Department of Chemical Biology, Max Planck Institute for Medical Research, Jahnstr. 29, 69120 Heidelberg, Germany.
  • Zirwes EA; Roche Pharma Research & Early Development, Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., 4070 Basel, Switzerland.
  • Guba W; Roche Pharma Research & Early Development, Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., 4070 Basel, Switzerland.
  • Grether U; Roche Pharma Research & Early Development, Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., 4070 Basel, Switzerland.
  • Frank JA; Roche Pharma Research & Early Development, Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., 4070 Basel, Switzerland.
  • Veprintsev DB; Department of Chemical Physiology & Biochemistry, Oregon Health & Science University, Portland, Oregon 97239-3098, United States.
  • Carreira EM; Vollum Institute, Oregon Health & Science University, Portland, Oregon 97239-3098, United States.
J Am Chem Soc ; 145(28): 15094-15108, 2023 07 19.
Article em En | MEDLINE | ID: mdl-37401816

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Transdução de Sinais / Corantes Fluorescentes Idioma: En Revista: J Am Chem Soc Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Suíça

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Transdução de Sinais / Corantes Fluorescentes Idioma: En Revista: J Am Chem Soc Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Suíça