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Kinetics, Thermodynamics, and Structural Effects of Quinoline-2-Carboxylates, Zinc-Binding Inhibitors of New Delhi Metallo-ß-lactamase-1 Re-sensitizing Multidrug-Resistant Bacteria for Carbapenems.
Jia, Yuwen; Schroeder, Barbara; Pfeifer, Yvonne; Fröhlich, Christopher; Deng, Lihua; Arkona, Christoph; Kuropka, Benno; Sticht, Jana; Ataka, Kenichi; Bergemann, Silke; Wolber, Gerhard; Nitsche, Christoph; Mielke, Martin; Leiros, Hanna-Kirsti S; Werner, Guido; Rademann, Jörg.
Afiliação
  • Jia Y; Institute of Pharmacy, Freie Universität Berlin, Königin-Luise-Str. 2+4, Berlin 14195, Germany.
  • Schroeder B; Institute of Pharmacy, Freie Universität Berlin, Königin-Luise-Str. 2+4, Berlin 14195, Germany.
  • Pfeifer Y; FG13 Nosocomial Pathogens and Antibiotic Resistances, Department of Infectious Diseases, Robert Koch Institute, Burgstraße 37, Wernigerode 38855, Germany.
  • Fröhlich C; Department of Chemistry, Faculty of Science and Technology, UiT The Arctic University of Norway, Tromsø 9037, Norway.
  • Deng L; Institute of Pharmacy, Freie Universität Berlin, Königin-Luise-Str. 2+4, Berlin 14195, Germany.
  • Arkona C; Institute of Pharmacy, Freie Universität Berlin, Königin-Luise-Str. 2+4, Berlin 14195, Germany.
  • Kuropka B; Core Facility BioSupraMol, Institute for Chemistry and Biochemistry, Freie Universität Berlin, Thielallee 63, Berlin 14195, Germany.
  • Sticht J; Core Facility BioSupraMol, Institute for Chemistry and Biochemistry, Freie Universität Berlin, Thielallee 63, Berlin 14195, Germany.
  • Ataka K; Department of Physics, Freie Universität Berlin, Arnimallee 14, Berlin 14195, Germany.
  • Bergemann S; Institute of Pharmacy, Freie Universität Berlin, Königin-Luise-Str. 2+4, Berlin 14195, Germany.
  • Wolber G; Institute of Pharmacy, Freie Universität Berlin, Königin-Luise-Str. 2+4, Berlin 14195, Germany.
  • Nitsche C; Research School of Chemistry, Australian National University, Canberra 2601, Australian Capital Territory, Australia.
  • Mielke M; Department of Infectious Diseases, Robert Koch Institute, Nordufer 20, Berlin 13353, Germany.
  • Leiros HS; Department of Chemistry, Faculty of Science and Technology, UiT The Arctic University of Norway, Tromsø 9037, Norway.
  • Werner G; FG13 Nosocomial Pathogens and Antibiotic Resistances, Department of Infectious Diseases, Robert Koch Institute, Burgstraße 37, Wernigerode 38855, Germany.
  • Rademann J; Institute of Pharmacy, Freie Universität Berlin, Königin-Luise-Str. 2+4, Berlin 14195, Germany.
J Med Chem ; 66(17): 11761-11791, 2023 09 14.
Article em En | MEDLINE | ID: mdl-37585683

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinolinas / Carbapenêmicos Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Alemanha

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinolinas / Carbapenêmicos Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Alemanha