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Fortuitous In Vitro Compound Degradation Produces a Tractable Hit against Mycobacterium tuberculosis Dethiobiotin Synthetase: A Cautionary Tale of What Goes In Does Not Always Come Out.
Salaemae, Wanisa; Thompson, Andrew P; Gaiser, Birgit I; Lee, Kwang Jun; Huxley, Michael T; Sumby, Christopher J; Polyak, Steven W; Abell, Andrew D; Bruning, John B; Wegener, Kate L.
Afiliação
  • Salaemae W; Biochemistry, Division of Health and Applied Sciences, Faculty of Science, Prince of Songkla University, Songkhla 90110, Thailand.
  • Thompson AP; Department of Molecular and Cellular Biology, School of Biological Sciences, University of Adelaide, Adelaide, SA 5005, Australia.
  • Gaiser BI; Centre for Nanoscale BioPhotonics (CNBP), School of Biological Sciences, University of Adelaide, Adelaide, SA 5005, Australia.
  • Lee KJ; Centre for Nanoscale BioPhotonics (CNBP), School of Biological Sciences, University of Adelaide, Adelaide, SA 5005, Australia.
  • Huxley MT; Institute of Photonics and Advanced Sensing (IPAS), School of Biological Sciences, University of Adelaide, Adelaide, SA 5005, Australia.
  • Sumby CJ; Department of Chemistry, School of Physics, Chemistry and Earth Sciences, University of Adelaide, Adelaide, SA 5005, Australia.
  • Polyak SW; Department of Chemistry, School of Physics, Chemistry and Earth Sciences, University of Adelaide, Adelaide, SA 5005, Australia.
  • Abell AD; Department of Molecular and Cellular Biology, School of Biological Sciences, University of Adelaide, Adelaide, SA 5005, Australia.
  • Bruning JB; Centre for Nanoscale BioPhotonics (CNBP), School of Biological Sciences, University of Adelaide, Adelaide, SA 5005, Australia.
  • Wegener KL; Institute of Photonics and Advanced Sensing (IPAS), School of Biological Sciences, University of Adelaide, Adelaide, SA 5005, Australia.
ACS Chem Biol ; 18(9): 1985-1992, 2023 09 15.
Article em En | MEDLINE | ID: mdl-37651626

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Carbono-Nitrogênio Ligases / Mycobacterium tuberculosis Tipo de estudo: Prognostic_studies Idioma: En Revista: ACS Chem Biol Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Tailândia

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Carbono-Nitrogênio Ligases / Mycobacterium tuberculosis Tipo de estudo: Prognostic_studies Idioma: En Revista: ACS Chem Biol Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Tailândia