Detalles de la búsqueda
1.
Synthesis, biological evaluation, and stability studies of raloxifene mono- and bis-sulfamates as dual-targeting agents.
Bioorg Med Chem
; 101: 117645, 2024 Mar 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-38401456
2.
Anti-proliferative activity of RIHMS-Qi-23 against MCF-7 breast cancer cell line is through inhibition of cell proliferation and senescence but not inhibition of targeted kinases.
BMC Cancer
; 23(1): 1053, 2023 Nov 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-37919708
3.
Design, synthesis, and biological evaluation of a new series of pyrazole derivatives: Discovery of potent and selective JNK3 kinase inhibitors.
Bioorg Med Chem
; 69: 116894, 2022 09 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-35764033
4.
Discovery of urease inhibitory effect of sulfamate derivatives: Biological and computational studies.
Bioorg Chem
; 119: 105545, 2022 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-34915286
5.
Evaluation of Substituted Pyrazole-Based Kinase Inhibitors in One Decade (2011-2020): Current Status and Future Prospects.
Molecules
; 27(1)2022 Jan 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-35011562
6.
A Review of HER4 (ErbB4) Kinase, Its Impact on Cancer, and Its Inhibitors.
Molecules
; 26(23)2021 Dec 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-34885957
7.
A new series of aryl sulfamate derivatives: Design, synthesis, and biological evaluation.
Bioorg Med Chem
; 28(8): 115406, 2020 04 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-32173116
8.
Evaluation of sulfonate and sulfamate derivatives possessing benzofuran or benzothiophene nucleus as inhibitors of nucleotide pyrophosphatases/phosphodiesterases and anticancer agents.
Bioorg Chem
; 104: 104305, 2020 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-33017718
9.
Synthesis, biological evaluation, and docking studies of new pyrazole-based thiourea and sulfonamide derivatives as inhibitors of nucleotide pyrophosphatase/phosphodiesterase.
Bioorg Chem
; 99: 103783, 2020 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-32224334
10.
Imidazothiazole-based potent inhibitors of V600E-B-RAF kinase with promising anti-melanoma activity: biological and computational studies.
J Enzyme Inhib Med Chem
; 35(1): 1712-1726, 2020 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-32962435
11.
Sulfonate and sulfamate derivatives possessing benzofuran or benzothiophene nucleus as potent carbonic anhydrase II/IX/XII inhibitors.
Bioorg Med Chem
; 27(17): 3889-3901, 2019 09 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-31345748
12.
Synthesis, biological evaluation, and molecular docking study of sulfonate derivatives as nucleotide pyrophosphatase/phosphodiesterase (NPP) inhibitors.
Bioorg Med Chem
; 27(13): 2741-2752, 2019 07 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-31088715
13.
Patients' Knowledge and Pharmacists' Practice Regarding the Long-Term Side Effects of Proton Pump Inhibitors; a Cross-sectional Study.
Arch Acad Emerg Med
; 12(1): e35, 2024.
Artículo
en Inglés
| MEDLINE | ID: mdl-38721447
14.
Design and discovery of urease and Helicobacter pylori inhibitors based on benzofuran/benzothiophene-sulfonate and sulfamate scaffolds for the treatment of ureolytic bacterial infections.
Int J Biol Macromol
; 271(Pt 1): 132502, 2024 May 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-38768915
15.
Design, synthesis, biological evaluation, and in silico studies of novel pyridopyridine derivatives as anticancer candidates targeting FMS kinase.
Eur J Med Chem
; 274: 116557, 2024 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-38850857
16.
FMS Kinase Inhibitors: Current Status and Future Prospects.
Med Res Rev
; 33(3): 599-636, 2013 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-22434539
17.
Discovery of olmesartan hexetil: a new potential prodrug of olmesartan.
Bioorg Med Chem Lett
; 23(5): 1347-50, 2013 Mar 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23347686
18.
Novel Anti-Acanthamoebic Activities of Irosustat and STX140 and Their Nanoformulations.
Antibiotics (Basel)
; 12(3)2023 Mar 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-36978428
19.
Promising drug candidates for the treatment of polycystic ovary syndrome (PCOS) as alternatives to the classical medication metformin.
Eur J Pharmacol
; 960: 176119, 2023 Dec 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-37852569
20.
Design and synthesis of novel anti-urease imidazothiazole derivatives with promising antibacterial activity against Helicobacter pylori.
PLoS One
; 18(6): e0286684, 2023.
Artículo
en Inglés
| MEDLINE | ID: mdl-37267378