Detalles de la búsqueda
1.
Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships.
J Enzyme Inhib Med Chem
; 38(1): 2201402, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37073528
2.
Phenylsulfonimide PPARα Antagonists Enhance Nrf2 Activation and Promote Oxidative Stress-Induced Apoptosis/Pyroptosis in MCF7 Breast Cancer Cells.
Int J Mol Sci
; 24(2)2023 Jan 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-36674831
3.
Antimicrobial and Antibiofilm Activities of Carvacrol, Amoxicillin and Salicylhydroxamic Acid Alone and in Combination vs. Helicobacter pylori: Towards a New Multi-Targeted Therapy.
Int J Mol Sci
; 24(5)2023 Feb 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-36901886
4.
Photoactivatable Heptamethine-Based Carbonic Anhydrase Inhibitors Leading to New Anti-Antibacterial Agents.
Int J Mol Sci
; 24(11)2023 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-37298561
5.
Kinetic Study on the Base-Catalyzed Imine-Enamine Tautomerism of a Chiral Biologically Active Isoxazoline Derivative by HPLC on Amylose Tris(3,5-dimethylphenylcarbamate) Chiral Stationary Phase.
Molecules
; 28(18)2023 Sep 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-37764294
6.
The kinesin Eg5 inhibitor K858 exerts antiproliferative and proapoptotic effects and attenuates the invasive potential of head and neck squamous carcinoma cells.
Invest New Drugs
; 40(3): 556-564, 2022 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-35312942
7.
Benzenesulfonamides with different rigidity-conferring linkers as carbonic anhydrase inhibitors: an insight into the antiproliferative effect on glioblastoma, pancreatic, and breast cancer cells.
J Enzyme Inhib Med Chem
; 37(1): 1857-1869, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-35768159
8.
Biological investigation of N-methyl thiosemicarbazones as antimicrobial agents and bacterial carbonic anhydrases inhibitors.
J Enzyme Inhib Med Chem
; 37(1): 986-993, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-35322729
9.
Natural and Synthetic Xanthone Derivatives Counteract Oxidative Stress via Nrf2 Modulation in Inflamed Human Macrophages.
Int J Mol Sci
; 23(21)2022 Nov 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-36362104
10.
Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies.
Int J Mol Sci
; 23(14)2022 Jul 19.
Artículo
en Inglés
| MEDLINE | ID: mdl-35887299
11.
Fisetin as a Senotherapeutic Agent: Biopharmaceutical Properties and Crosstalk between Cell Senescence and Neuroprotection.
Molecules
; 27(3)2022 Jan 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-35164003
12.
Negative Modulation of the Angiogenic Cascade Induced by Allosteric Kinesin Eg5 Inhibitors in a Gastric Adenocarcinoma In Vitro Model.
Molecules
; 27(3)2022 Jan 31.
Artículo
en Inglés
| MEDLINE | ID: mdl-35164221
13.
Coumarin-Based Dual Inhibitors of Human Carbonic Anhydrases and Monoamine Oxidases Featuring Amino Acyl and (Pseudo)-Dipeptidyl Appendages: In Vitro and Computational Studies.
Molecules
; 27(22)2022 Nov 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-36431985
14.
Resveratrol Analogues as Dual Inhibitors of Monoamine Oxidase B and Carbonic Anhydrase VII: A New Multi-Target Combination for Neurodegenerative Diseases?
Molecules
; 27(22)2022 Nov 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-36431918
15.
Design, Synthesis and Biological Assessment of Rhodanine-Linked Benzenesulfonamide Derivatives as Selective and Potent Human Carbonic Anhydrase Inhibitors.
Molecules
; 27(22)2022 Nov 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-36432129
16.
Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase.
J Enzyme Inhib Med Chem
; 36(1): 561-580, 2021 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-33615947
17.
New azolyl-derivatives as multitargeting agents against breast cancer and fungal infections: synthesis, biological evaluation and docking study.
J Enzyme Inhib Med Chem
; 36(1): 1632-1645, 2021 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-34289751
18.
Selective Inhibition of Helicobacter pylori Carbonic Anhydrases by Carvacrol and Thymol Could Impair Biofilm Production and the Release of Outer Membrane Vesicles.
Int J Mol Sci
; 22(21)2021 Oct 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-34769015
19.
Novel Biologically Active Molecules, Biomaterials, and Nanoparticles for Microbial Biofilm Control in Human Medicine.
Molecules
; 26(9)2021 May 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-34067036
20.
Amine- and Amino Acid-Based Compounds as Carbonic Anhydrase Activators.
Molecules
; 26(23)2021 Dec 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-34885917