Detalles de la búsqueda
1.
Boron-containing carbonic anhydrases inhibitors.
Bioorg Chem
; 143: 106976, 2024 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-38000350
2.
Coumarins-lipophilic cations conjugates: Efficient mitocans targeting carbonic anhydrases.
Bioorg Chem
; 145: 107168, 2024 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-38354500
3.
Development of a multi-targeted chemotherapeutic approach based on G-quadruplex stabilisation and carbonic anhydrase inhibition.
J Enzyme Inhib Med Chem
; 39(1): 2366236, 2024 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-38905127
4.
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains.
Int J Mol Sci
; 25(5)2024 Feb 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-38473830
5.
Leveraging SARS-CoV-2 Main Protease (Mpro) for COVID-19 Mitigation with Selenium-Based Inhibitors.
Int J Mol Sci
; 25(2)2024 Jan 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-38256046
6.
Design and synthesis of sulfonamides incorporating a biotin moiety: Carbonic anhydrase inhibitory effects, antiproliferative activity and molecular modeling studies.
Bioorg Med Chem
; 94: 117467, 2023 Oct 30.
Artículo
en Inglés
| MEDLINE | ID: mdl-37722299
7.
1,2,3-Benzoxathiazine-2,2-dioxides - effective inhibitors of human carbonic anhydrases.
J Enzyme Inhib Med Chem
; 38(1): 225-238, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36373195
8.
3H-1,2-Benzoxaphosphepine 2-oxides as selective inhibitors of carbonic anhydrase IX and XII.
J Enzyme Inhib Med Chem
; 38(1): 216-224, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36377338
9.
Diversely N-substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N-nitrosulfonamides.
J Enzyme Inhib Med Chem
; 38(1): 2178430, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36798036
10.
Aryl derivatives of 3H-1,2-benzoxaphosphepine 2-oxides as inhibitors of cancer-related carbonic anhydrase isoforms IX and XII.
J Enzyme Inhib Med Chem
; 38(1): 2249267, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37655449
11.
Antihistamines, phenothiazine-based antipsychotics, and tricyclic antidepressants potently activate pharmacologically relevant human carbonic anhydrase isoforms II and VII.
J Enzyme Inhib Med Chem
; 38(1): 2188147, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36912265
12.
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors.
J Enzyme Inhib Med Chem
; 38(1): 2202360, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37092262
13.
Derivatives of 4-methyl-1,2,3-benzoxathiazine 2,2-dioxide as selective inhibitors of human carbonic anhydrases IX and XII over the cytosolic isoforms I and II.
J Enzyme Inhib Med Chem
; 38(1): 2170370, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36718988
14.
New isoxazolidinyl-based N-alkylethanolamines as new activators of human brain carbonic anhydrases.
J Enzyme Inhib Med Chem
; 38(1): 2164574, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36630083
15.
Discovery of new 6-ureido/amidocoumarins as highly potent and selective inhibitors for the tumour-relevant carbonic anhydrases IX and XII.
J Enzyme Inhib Med Chem
; 38(1): 2154603, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36728712
16.
Development of novel anilinoquinazoline-based carboxylic acids as non-classical carbonic anhydrase IX and XII inhibitors.
J Enzyme Inhib Med Chem
; 38(1): 2191163, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36942698
17.
Design, synthesis, and biological investigation of selective human carbonic anhydrase II, IX, and XII inhibitors using 7-aryl/heteroaryl triazolopyrimidines bearing a sulfanilamide scaffold.
J Enzyme Inhib Med Chem
; 38(1): 2270180, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37850364
18.
Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates.
J Enzyme Inhib Med Chem
; 38(1): 2284119, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37994421
19.
Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights.
J Enzyme Inhib Med Chem
; 38(1): 2201407, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37078173
20.
The role of carbonic anhydrases in extinction of contextual fear memory.
Proc Natl Acad Sci U S A
; 117(27): 16000-16008, 2020 07 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-32571910