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1.
Diastereoselective synthesis of cyclic tetrapeptide pseudoxylallemycin A illuminates the impact of base during macrolactamization.
Org Biomol Chem
; 21(5): 1056-1069, 2023 02 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-36628602
2.
A general, enantioselective synthesis of N-alkyl terminal aziridines and C2-functionalized azetidines via organocatalysis.
Tetrahedron Lett
; 56(10): 1276-1279, 2015 Mar 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-26834294
3.
Regulation of phospholipase D activity and phosphatidic acid production after purinergic (P2Y6) receptor stimulation.
J Biol Chem
; 288(28): 20477-87, 2013 Jul 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-23723068
4.
Further evaluation of novel structural modifications to scaffolds that engender PLD isoform selective inhibition.
Bioorg Med Chem Lett
; 24(24): 5553-5557, 2014 Dec 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-25466173
5.
A general, enantioselective synthesis of ß- and γ-fluoroamines.
Tetrahedron Lett
; 54(28): 3627-3629, 2013 Jul 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-24039308
6.
Scalable and Chromatography-Free Synthesis of Efflux Pump Inhibitor Phenylalanine Arginine ß-Naphthylamide for Its Validation in Wild-Type Bacterial Strains.
ChemMedChem
; 18(14): e202300128, 2023 07 17.
Artículo
en Inglés
| MEDLINE | ID: mdl-37126222
7.
Enantioselective synthesis of C2-functionalized, N-protected morpholines and orthogonally N,N'-protected piperazines via organocatalysis.
Tetrahedron Lett
; 53(13): 1539-1542, 2012 Mar 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-22919116
8.
Synthesis and Characterization of Functionalized Amino Dihydropyrimidines Toward the Analysis of their Antibacterial Structure-Activity Relationships and Mechanism of Action.
ACS Omega
; 7(42): 37907-37916, 2022 Oct 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-36312355
9.
Design, Synthesis, and Biochemical Characterization of Non-Native Antagonists of the Pseudomonas aeruginosa Quorum Sensing Receptor LasR with Nanomolar IC50 Values.
ACS Infect Dis
; 6(4): 649-661, 2020 04 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-32037806
10.
Structural and Biochemical Studies of Non-native Agonists of the LasR Quorum-Sensing Receptor Reveal an L3 Loop "Out" Conformation for LasR.
Cell Chem Biol
; 25(9): 1128-1139.e3, 2018 09 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-30033130
11.
Structure-Based Design and Biological Evaluation of Triphenyl Scaffold-Based Hybrid Compounds as Hydrolytically Stable Modulators of a LuxR-Type Quorum Sensing Receptor.
ACS Infect Dis
; 2(1): 32-38, 2016 Jan 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-26807436
12.
Discovery of desketoraloxifene analogues as inhibitors of mammalian, Pseudomonas aeruginosa, and NAPE phospholipase D enzymes.
ACS Chem Biol
; 10(2): 421-32, 2015 Feb 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-25384256
13.
Discovery of a highly selective PLD2 inhibitor (ML395): a new probe with improved physiochemical properties and broad-spectrum antiviral activity against influenza strains.
ChemMedChem
; 9(12): 2633-7, 2014 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-25210004
14.
Development of dual PLD1/2 and PLD2 selective inhibitors from a common 1,3,8-Triazaspiro[4.5]decane Core: discovery of Ml298 and Ml299 that decrease invasive migration in U87-MG glioblastoma cells.
J Med Chem
; 56(6): 2695-9, 2013 Mar 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-23445448
15.
A general, enantioselective synthesis of protected morpholines and piperazines.
Org Lett
; 14(11): 2910-3, 2012 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-22616979
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