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1.
Discovery and Development of TMPRSS6 Inhibitors Modulating Hepcidin Levels in Human Hepatocytes.
Cell Chem Biol
; 26(11): 1559-1572.e9, 2019 11 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-31543462
2.
Identification via a Parallel Hit Progression Strategy of Improved Small Molecule Inhibitors of the Malaria Purine Uptake Transporter that Inhibit Plasmodium falciparum Parasite Proliferation.
ACS Infect Dis
; 5(10): 1738-1753, 2019 10 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-31373203
3.
Inhibitors of LexA Autoproteolysis and the Bacterial SOS Response Discovered by an Academic-Industry Partnership.
ACS Infect Dis
; 4(3): 349-359, 2018 03 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-29275629
4.
A High-Content Imaging Screen for Cellular Regulators of ß-Catenin Protein Abundance.
J Biomol Screen
; 21(3): 260-8, 2016 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-26656867
5.
Cell-Based Selection Expands the Utility of DNA-Encoded Small-Molecule Library Technology to Cell Surface Drug Targets: Identification of Novel Antagonists of the NK3 Tachykinin Receptor.
ACS Comb Sci
; 17(12): 722-31, 2015 Dec 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-26562224
6.
Nanomolar inhibitors of Staphylococcus aureus methionyl tRNA synthetase with potent antibacterial activity against gram-positive pathogens.
J Med Chem
; 45(10): 1959-62, 2002 May 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-11985462
7.
Single-molecule detection technologies in miniaturized high-throughput screening: fluorescence intensity distribution analysis.
J Biomol Screen
; 8(1): 19-33, 2003 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-12854995
8.
A standard operating procedure for assessing liquid handler performance in high-throughput screening.
J Biomol Screen
; 7(6): 554-69, 2002 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-14599354
9.
A novel approach applying a chemical biology strategy in phenotypic screening reveals pathway-selective regulators of histone 3 K27 tri-methylation.
Mol Biosyst
; 10(2): 251-7, 2014 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-24257700
10.
Development of phenotypic screening assays for γ-globin induction using primary human bone marrow day 7 erythroid progenitor cells.
J Biomol Screen
; 18(10): 1212-22, 2013 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-24163393
11.
Perspectives on the discovery of small-molecule modulators for epigenetic processes.
J Biomol Screen
; 17(5): 555-71, 2012 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-22392809
12.
Development and validation of reagents and assays for EZH2 peptide and nucleosome high-throughput screens.
J Biomol Screen
; 17(10): 1279-92, 2012 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-22904200
13.
Conformational restriction of methionyl tRNA synthetase inhibitors leading to analogues with potent inhibition and excellent gram-positive antibacterial activity.
Bioorg Med Chem Lett
; 13(7): 1265-8, 2003 Apr 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-12657260
14.
The antimicrobial natural product chuangxinmycin and some synthetic analogues are potent and selective inhibitors of bacterial tryptophanyl tRNA synthetase.
Bioorg Med Chem Lett
; 12(21): 3171-4, 2002 Nov 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-12372526
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