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From Drug Screening to Target Deconvolution: a Target-Based Drug Discovery Pipeline Using Leishmania Casein Kinase 1 Isoform 2 To Identify Compounds with Antileishmanial Activity.
Durieu, Emilie; Prina, Eric; Leclercq, Olivier; Oumata, Nassima; Gaboriaud-Kolar, Nicolas; Vougogiannopoulou, Konstantina; Aulner, Nathalie; Defontaine, Audrey; No, Joo Hwan; Ruchaud, Sandrine; Skaltsounis, Alexios-Leandros; Galons, Hervé; Späth, Gerald F; Meijer, Laurent; Rachidi, Najma.
Afiliación
  • Durieu E; Sorbonne Universités, UPMC Université de Paris 06, CNRS USR3151, Protein Phosphorylation and Human Diseases, Station Biologique, Roscoff, France.
  • Prina E; Institut Pasteur, Laboratoire d'Immunophysiologie et Parasitisme, Paris, France.
  • Leclercq O; Institut Pasteur and INSERM U1201, Unité de Parasitologie moléculaire et Signalisation, Paris, France.
  • Oumata N; ManRos Therapeutics, Centre de Perharidy, Roscoff, France.
  • Gaboriaud-Kolar N; Department of Pharmacognosy and Natural Products Chemistry, School of Pharmacy, University of Athens, Athens, Greece.
  • Vougogiannopoulou K; Department of Pharmacognosy and Natural Products Chemistry, School of Pharmacy, University of Athens, Athens, Greece.
  • Aulner N; Institut Pasteur, Imagopole, Paris, France.
  • Defontaine A; Sorbonne Universités, UPMC Université de Paris 06, CNRS USR3151, Protein Phosphorylation and Human Diseases, Station Biologique, Roscoff, France.
  • No JH; Institut Pasteur Korea, Leishmania Research Laboratory, Seongnam-si, Republic of Korea.
  • Ruchaud S; Sorbonne Universités, UPMC Université de Paris 06, CNRS USR3151, Protein Phosphorylation and Human Diseases, Station Biologique, Roscoff, France.
  • Skaltsounis AL; Department of Pharmacognosy and Natural Products Chemistry, School of Pharmacy, University of Athens, Athens, Greece.
  • Galons H; Université Paris-Descartes, Laboratoire de Chimie Organique 2, INSERM U 648, Paris, France.
  • Späth GF; Institut Pasteur and INSERM U1201, Unité de Parasitologie moléculaire et Signalisation, Paris, France.
  • Meijer L; Sorbonne Universités, UPMC Université de Paris 06, CNRS USR3151, Protein Phosphorylation and Human Diseases, Station Biologique, Roscoff, France.
  • Rachidi N; Sorbonne Universités, UPMC Université de Paris 06, CNRS USR3151, Protein Phosphorylation and Human Diseases, Station Biologique, Roscoff, France najma.rachidi@pasteur.fr.
Antimicrob Agents Chemother ; 60(5): 2822-33, 2016 05.
Article en En | MEDLINE | ID: mdl-26902771

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Leishmania / Antiprotozoarios Tipo de estudio: Diagnostic_studies / Screening_studies Límite: Animals / Humans Idioma: En Revista: Antimicrob Agents Chemother Año: 2016 Tipo del documento: Article País de afiliación: Francia

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Leishmania / Antiprotozoarios Tipo de estudio: Diagnostic_studies / Screening_studies Límite: Animals / Humans Idioma: En Revista: Antimicrob Agents Chemother Año: 2016 Tipo del documento: Article País de afiliación: Francia