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RVX-297- a novel BD2 selective inhibitor of BET bromodomains.
Kharenko, Olesya A; Gesner, Emily M; Patel, Reena G; Norek, Karen; White, Andre; Fontano, Eric; Suto, Robert K; Young, Peter R; McLure, Kevin G; Hansen, Henrik C.
Afiliación
  • Kharenko OA; Zenith Epigenetics, Suite 300, 4820 Richard Road SW, Calgary, Alberta, T3E 6L1, Canada. Electronic address: olesya@zenithepigenetics.com.
  • Gesner EM; Zenith Epigenetics, Suite 300, 4820 Richard Road SW, Calgary, Alberta, T3E 6L1, Canada.
  • Patel RG; Zenith Epigenetics, Suite 300, 4820 Richard Road SW, Calgary, Alberta, T3E 6L1, Canada.
  • Norek K; Zenith Epigenetics, Suite 300, 4820 Richard Road SW, Calgary, Alberta, T3E 6L1, Canada.
  • White A; Xtal BioStructures, Inc., 12 Michigan Dr., Natick, MA 01760, USA.
  • Fontano E; Xtal BioStructures, Inc., 12 Michigan Dr., Natick, MA 01760, USA.
  • Suto RK; Xtal BioStructures, Inc., 12 Michigan Dr., Natick, MA 01760, USA.
  • Young PR; Zenith Epigenetics, Suite 300, 4820 Richard Road SW, Calgary, Alberta, T3E 6L1, Canada.
  • McLure KG; Zenith Epigenetics, Suite 300, 4820 Richard Road SW, Calgary, Alberta, T3E 6L1, Canada.
  • Hansen HC; Zenith Epigenetics, Suite 300, 4820 Richard Road SW, Calgary, Alberta, T3E 6L1, Canada.
Biochem Biophys Res Commun ; 477(1): 62-67, 2016 08 12.
Article en En | MEDLINE | ID: mdl-27282480

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Factores de Transcripción / Quinazolinonas Idioma: En Revista: Biochem Biophys Res Commun Año: 2016 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Factores de Transcripción / Quinazolinonas Idioma: En Revista: Biochem Biophys Res Commun Año: 2016 Tipo del documento: Article