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A new nitrobenzoxadiazole-based GSTP1-1 inhibitor with a previously unheard of mechanism of action and high stability.
Fulci, Chiara; Rotili, Dante; De Luca, Anastasia; Stella, Lorenzo; Morozzo Della Rocca, Blasco; Forgione, Mariantonietta; Di Paolo, Veronica; Mai, Antonello; Falconi, Mattia; Quintieri, Luigi; Caccuri, Anna M.
Afiliación
  • Fulci C; a Department of Experimental Medicine and Surgery , University of Tor Vergata , Rome , Italy.
  • Rotili D; b Department of Drug Chemistry and Technologies , University of Rome "Sapienza" , Rome , Italy.
  • De Luca A; a Department of Experimental Medicine and Surgery , University of Tor Vergata , Rome , Italy.
  • Stella L; c Department of Chemical Sciences and Technologies.
  • Morozzo Della Rocca B; d Department of Biology , University of Tor Vergata , Rome , Italy.
  • Forgione M; b Department of Drug Chemistry and Technologies , University of Rome "Sapienza" , Rome , Italy.
  • Di Paolo V; e Department of Pharmaceutical and Pharmacological Sciences , University of Padova , Padova , Italy.
  • Mai A; b Department of Drug Chemistry and Technologies , University of Rome "Sapienza" , Rome , Italy.
  • Falconi M; f Pasteur Institute, Cenci Bolognetti Foundation, University of Rome "La Sapienza" , Rome , Italy.
  • Quintieri L; d Department of Biology , University of Tor Vergata , Rome , Italy.
  • Caccuri AM; e Department of Pharmaceutical and Pharmacological Sciences , University of Padova , Padova , Italy.
J Enzyme Inhib Med Chem ; 32(1): 240-247, 2017 Dec.
Article en En | MEDLINE | ID: mdl-28097896

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Oxazoles / Inhibidores Enzimáticos / Gutatión-S-Transferasa pi Límite: Humans Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: Italia

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Oxazoles / Inhibidores Enzimáticos / Gutatión-S-Transferasa pi Límite: Humans Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: Italia