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New N-phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity.
Durcik, Martina; Lovison, Denise; Skok, Ziga; Durante Cruz, Cristina; Tammela, Päivi; Tomasic, Tihomir; Benedetto Tiz, Davide; Draskovits, Gábor; Nyerges, Ákos; Pál, Csaba; Ilas, Janez; Peterlin Masic, Lucija; Kikelj, Danijel; Zidar, Nace.
Afiliación
  • Durcik M; Faculty of Pharmacy, University of Ljubljana, Askerceva cesta 7, 1000, Ljubljana, Slovenia.
  • Lovison D; Faculty of Pharmacy, University of Ljubljana, Askerceva cesta 7, 1000, Ljubljana, Slovenia.
  • Skok Z; Faculty of Pharmacy, University of Ljubljana, Askerceva cesta 7, 1000, Ljubljana, Slovenia.
  • Durante Cruz C; Drug Research Program, Division of Pharmaceutical Biosciences, Faculty of Pharmacy, University of Helsinki, P.O. Box 56 (Viikinkaari 5 E), 00014, Helsinki, Finland.
  • Tammela P; Drug Research Program, Division of Pharmaceutical Biosciences, Faculty of Pharmacy, University of Helsinki, P.O. Box 56 (Viikinkaari 5 E), 00014, Helsinki, Finland.
  • Tomasic T; Faculty of Pharmacy, University of Ljubljana, Askerceva cesta 7, 1000, Ljubljana, Slovenia.
  • Benedetto Tiz D; Faculty of Pharmacy, University of Ljubljana, Askerceva cesta 7, 1000, Ljubljana, Slovenia.
  • Draskovits G; Synthetic and Systems Biology Unit, Institute of Biochemistry, Biological Research Centre of the Hungarian Academy of Sciences, Szeged, H-6726, Hungary.
  • Nyerges Á; Synthetic and Systems Biology Unit, Institute of Biochemistry, Biological Research Centre of the Hungarian Academy of Sciences, Szeged, H-6726, Hungary.
  • Pál C; Synthetic and Systems Biology Unit, Institute of Biochemistry, Biological Research Centre of the Hungarian Academy of Sciences, Szeged, H-6726, Hungary.
  • Ilas J; Faculty of Pharmacy, University of Ljubljana, Askerceva cesta 7, 1000, Ljubljana, Slovenia.
  • Peterlin Masic L; Faculty of Pharmacy, University of Ljubljana, Askerceva cesta 7, 1000, Ljubljana, Slovenia.
  • Kikelj D; Faculty of Pharmacy, University of Ljubljana, Askerceva cesta 7, 1000, Ljubljana, Slovenia.
  • Zidar N; Faculty of Pharmacy, University of Ljubljana, Askerceva cesta 7, 1000, Ljubljana, Slovenia. Electronic address: nace.zidar@ffa.uni-lj.si.
Eur J Med Chem ; 154: 117-132, 2018 Jun 25.
Article en En | MEDLINE | ID: mdl-29778894

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Pirroles / Staphylococcus aureus / Enterococcus faecalis / Girasa de ADN / Escherichia coli / Inhibidores de Topoisomerasa II / Amidas / Antibacterianos Idioma: En Revista: Eur J Med Chem Año: 2018 Tipo del documento: Article País de afiliación: Eslovenia

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Pirroles / Staphylococcus aureus / Enterococcus faecalis / Girasa de ADN / Escherichia coli / Inhibidores de Topoisomerasa II / Amidas / Antibacterianos Idioma: En Revista: Eur J Med Chem Año: 2018 Tipo del documento: Article País de afiliación: Eslovenia