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Cholesteryl ester transfer protein (CETP) inhibitors based on cyclic urea, bicyclic urea and bicyclic sulfamide cores.
Liu, Jian; Shao, Patrick P; Guiadeen, Deodial; Krikorian, Arto; Sun, Wanying; Deng, Qiaolin; Cumiskey, Anne-Marie; Duffy, Ruth A; Murphy, Beth A; Mitra, Kaushik; Johns, Douglas G; Duffy, Joseph L; Vachal, Petr.
Afiliación
  • Liu J; Discovery Chemistry, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, NJ 07033, USA. Electronic address: jianliu9600@gmail.com.
  • Shao PP; Discovery Chemistry, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, NJ 07033, USA.
  • Guiadeen D; Discovery Chemistry, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, NJ 07033, USA.
  • Krikorian A; Discovery Chemistry, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, NJ 07033, USA.
  • Sun W; Discovery Chemistry, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, NJ 07033, USA.
  • Deng Q; Discovery Chemistry, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, NJ 07033, USA.
  • Cumiskey AM; Discovery Biology, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, NJ 07033, USA.
  • Duffy RA; Discovery Biology, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, NJ 07033, USA.
  • Murphy BA; Discovery Biology, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, NJ 07033, USA.
  • Mitra K; Department of Drug Metabolism and Pharmacokinetics, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, NJ 07033, USA.
  • Johns DG; Discovery Biology, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, NJ 07033, USA.
  • Duffy JL; Discovery Chemistry, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, NJ 07033, USA.
  • Vachal P; Discovery Chemistry, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, NJ 07033, USA.
Bioorg Med Chem Lett ; 32: 127668, 2021 01 15.
Article en En | MEDLINE | ID: mdl-33161125

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Sulfonamidas / Urea / Compuestos Bicíclicos con Puentes / Proteínas de Transferencia de Ésteres de Colesterol / Anticolesterolemiantes Límite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2021 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Sulfonamidas / Urea / Compuestos Bicíclicos con Puentes / Proteínas de Transferencia de Ésteres de Colesterol / Anticolesterolemiantes Límite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2021 Tipo del documento: Article