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Structural determinants for subnanomolar inhibition of the secreted aspartic protease Sapp1p from Candida parapsilosis.
Dostál, Jirí; Brynda, Jirí; Vanková, Lucie; Zia, Syeda Rehana; Pichová, Iva; Heidingsfeld, Olga; Lepsík, Martin.
Afiliación
  • Dostál J; Institute of Organic Chemistry and Biochemistry, Czech Academy of Sciences, Prague, Czech Republic.
  • Brynda J; Institute of Organic Chemistry and Biochemistry, Czech Academy of Sciences, Prague, Czech Republic.
  • Vanková L; Laboratory of Ligand Engineering, Institute of Biotechnology, Czech Academy of Sciences, v.v.i., BIOCEV Research Center, Vestec, Czech Republic.
  • Zia SR; Department of Chemistry, University of Karachi, Karachi, Pakistan.
  • Pichová I; Institute of Organic Chemistry and Biochemistry, Czech Academy of Sciences, Prague, Czech Republic.
  • Heidingsfeld O; Institute of Organic Chemistry and Biochemistry, Czech Academy of Sciences, Prague, Czech Republic.
  • Lepsík M; Department of Biochemistry, Faculty of Science, Charles University in Prague, Prague, Czech Republic.
J Enzyme Inhib Med Chem ; 36(1): 914-921, 2021 Dec.
Article en En | MEDLINE | ID: mdl-33843395

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Inhibidores de Proteasas / Proteínas Fúngicas / Ácido Aspártico Endopeptidasas / Peptidomiméticos / Candida parapsilosis Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2021 Tipo del documento: Article País de afiliación: República Checa

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Inhibidores de Proteasas / Proteínas Fúngicas / Ácido Aspártico Endopeptidasas / Peptidomiméticos / Candida parapsilosis Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2021 Tipo del documento: Article País de afiliación: República Checa