Design and characterisation of piperazine-benzofuran integrated dinitrobenzenesulfonamide as <i>Mycobacterium tuberculosis</i> H37Rv strain inhibitors.

Murthy, Vallabhaneni S; Tamboli, Yasinalli; Krishna, Vagolu Siva; Sriram, Dharmarajan; Akber Ansari, Siddique; Alarfaj, Abdullah A; Hirad, Abdurahman H; Vijayakumar, Vijayaparthasarathi

Design and characterisation of piperazine-benzofuran integrated dinitrobenzenesulfonamide as Mycobacterium tuberculosis H37Rv strain inhibitors.

Murthy, Vallabhaneni S; Tamboli, Yasinalli; Krishna, Vagolu Siva; Sriram, Dharmarajan; Akber Ansari, Siddique; Alarfaj, Abdullah A; Hirad, Abdurahman H; Vijayakumar, Vijayaparthasarathi.

Afiliación

Murthy VS; Centre for Organic and Medicinal Chemistry, Department of Chemistry, School of Advanced Sciences, VIT University, Vellore, India.
Tamboli Y; Centre for Organic and Medicinal Chemistry, Department of Chemistry, School of Advanced Sciences, VIT University, Vellore, India.
Krishna VS; Medicinal Chemistry and Antimycobacterial Research Laboratory, Pharmacy Group, Birla Institute of Technology and Science, Pilani, Hyderabad Campus, Hyderabad, India.
Sriram D; Medicinal Chemistry and Antimycobacterial Research Laboratory, Pharmacy Group, Birla Institute of Technology and Science, Pilani, Hyderabad Campus, Hyderabad, India.
Akber Ansari S; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh, Saudi Arabia.
Alarfaj AA; Department of Botany and Microbiology, College of Science, King Saud University, Riyadh, Saudi Arabia.
Hirad AH; Department of Botany and Microbiology, College of Science, King Saud University, Riyadh, Saudi Arabia.
Vijayakumar V; Centre for Organic and Medicinal Chemistry, Department of Chemistry, School of Advanced Sciences, VIT University, Vellore, India.

J Enzyme Inhib Med Chem ; 36(1): 1751-1759, 2021 Dec.

Article en En | MEDLINE | ID: mdl-34325595

Asunto(s)

Antituberculosos/química; Antituberculosos/farmacología; Bencenosulfonatos/química; Benzofuranos/química; Diseño de Fármacos; Mycobacterium tuberculosis/efectos de los fármacos; Piperazina/química; Amidas/química; Línea Celular Tumoral; Ensayos de Selección de Medicamentos Antitumorales; Humanos; Pruebas de Sensibilidad Microbiana; Simulación del Acoplamiento Molecular; Análisis Espectral/métodos

Palabras clave

2,4-dinitrobenzene sulphonamide; Piperazine-benzofuran; amino acid; anti-TB; hybridisation

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Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Bencenosulfonatos / Benzofuranos / Diseño de Fármacos / Piperazina / Mycobacterium tuberculosis / Antituberculosos Límite: Humans Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2021 Tipo del documento: Article País de afiliación: India

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