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Design, Synthesis, and Biological Activity of New CB2 Receptor Ligands: from Orthosteric and Allosteric Modulators to Dualsteric/Bitopic Ligands.
Gado, Francesca; Ferrisi, Rebecca; Polini, Beatrice; Mohamed, Kawthar A; Ricardi, Caterina; Lucarini, Elena; Carpi, Sara; Domenichini, Federica; Stevenson, Lesley A; Rapposelli, Simona; Saccomanni, Giuseppe; Nieri, Paola; Ortore, Gabriella; Pertwee, Roger G; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Chiellini, Grazia; Laprairie, Robert B; Manera, Clementina.
Afiliación
  • Gado F; Department of Pharmacy, University of Pisa, Pisa 56126, Italy.
  • Ferrisi R; Department of Pharmacy, University of Pisa, Pisa 56126, Italy.
  • Polini B; Department of Pharmacy, University of Pisa, Pisa 56126, Italy.
  • Mohamed KA; Department of Pathology, University of Pisa, Pisa 56126, Italy.
  • Ricardi C; College of Pharmacy and Nutrition, University of Saskatchewan, Saskatoon SK S7N 5E5, Canada.
  • Lucarini E; Department of Pathology, University of Pisa, Pisa 56126, Italy.
  • Carpi S; Department of Neuroscience, Psychology, Drug Research and Child Health, Section of Pharmacology and Toxicology, University of Florence, Florence 50139, Italy.
  • Domenichini F; Department of Pharmacy, University of Pisa, Pisa 56126, Italy.
  • Stevenson LA; NEST, Istituto Nanoscienze-CNR and Scuola Normale Superiore, Piazza San Silvestro, Pisa 56126, Italy.
  • Rapposelli S; Department of Pharmacy, University of Pisa, Pisa 56126, Italy.
  • Saccomanni G; Institute of Medical Sciences, University of Aberdeen, Aberdeen AB25 2ZD, Scotland, U.K.
  • Nieri P; Department of Pharmacy, University of Pisa, Pisa 56126, Italy.
  • Ortore G; CISUP, Centre for Instrumentation Sharing Pisa University, Lungarno Pacinotti 43, Pisa 56126, Italy.
  • Pertwee RG; Department of Pharmacy, University of Pisa, Pisa 56126, Italy.
  • Ghelardini C; Department of Pharmacy, University of Pisa, Pisa 56126, Italy.
  • Di Cesare Mannelli L; Department of Pharmacy, University of Pisa, Pisa 56126, Italy.
  • Chiellini G; Institute of Medical Sciences, University of Aberdeen, Aberdeen AB25 2ZD, Scotland, U.K.
  • Laprairie RB; Department of Neuroscience, Psychology, Drug Research and Child Health, Section of Pharmacology and Toxicology, University of Florence, Florence 50139, Italy.
  • Manera C; Department of Neuroscience, Psychology, Drug Research and Child Health, Section of Pharmacology and Toxicology, University of Florence, Florence 50139, Italy.
J Med Chem ; 65(14): 9918-9938, 2022 07 28.
Article en En | MEDLINE | ID: mdl-35849804

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Receptores Acoplados a Proteínas G / Receptor Cannabinoide CB2 Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2022 Tipo del documento: Article País de afiliación: Italia

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Receptores Acoplados a Proteínas G / Receptor Cannabinoide CB2 Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2022 Tipo del documento: Article País de afiliación: Italia