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Imidazo[1,2-a]Pyridine Derivatives as Novel Dual-Target Inhibitors of ABCB1 and ABCG2 for Reversing Multidrug Resistance.
Li, Hui; Zhang, Sheng-Lie; Jia, Yan-Han; Li, Qian; Feng, Zi-Wen; Zhang, Shi-Duo; Zheng, Wei; Zhou, Ye-Ling; Li, Lin-Lin; Liu, Xue-Chun; Chen, Ya-Qiong; Peng, Hui; You, Qi-Dong; Xu, Xiao-Li.
Afiliación
  • Li H; State Key Laboratory of Natural Medicines, and Jiang Su Key Laboratory of Drug Design and Optimization, China Pharmaceutical University, Nanjing 210009, China.
  • Zhang SL; Department of Medicinal Chemistry, School of Pharmacy, China Pharmaceutical University, Nanjing 210009, China.
  • Jia YH; State Key Laboratory of Natural Medicines, and Jiang Su Key Laboratory of Drug Design and Optimization, China Pharmaceutical University, Nanjing 210009, China.
  • Li Q; Department of Medicinal Chemistry, School of Pharmacy, China Pharmaceutical University, Nanjing 210009, China.
  • Feng ZW; Department of Operational Medicine, Tianjin Institute of Environmental & Operational Medicine, Tianjin 300050, China.
  • Zhang SD; State Key Laboratory of Natural Medicines, and Jiang Su Key Laboratory of Drug Design and Optimization, China Pharmaceutical University, Nanjing 210009, China.
  • Zheng W; Department of Medicinal Chemistry, School of Pharmacy, China Pharmaceutical University, Nanjing 210009, China.
  • Zhou YL; State Key Laboratory of Natural Medicines, and Jiang Su Key Laboratory of Drug Design and Optimization, China Pharmaceutical University, Nanjing 210009, China.
  • Li LL; Department of Medicinal Chemistry, School of Pharmacy, China Pharmaceutical University, Nanjing 210009, China.
  • Liu XC; State Key Laboratory of Natural Medicines, and Jiang Su Key Laboratory of Drug Design and Optimization, China Pharmaceutical University, Nanjing 210009, China.
  • Chen YQ; Department of Medicinal Chemistry, School of Pharmacy, China Pharmaceutical University, Nanjing 210009, China.
  • Peng H; State Key Laboratory of Natural Medicines, and Jiang Su Key Laboratory of Drug Design and Optimization, China Pharmaceutical University, Nanjing 210009, China.
  • You QD; Department of Medicinal Chemistry, School of Pharmacy, China Pharmaceutical University, Nanjing 210009, China.
  • Xu XL; State Key Laboratory of Natural Medicines, and Jiang Su Key Laboratory of Drug Design and Optimization, China Pharmaceutical University, Nanjing 210009, China.
J Med Chem ; 66(4): 2804-2831, 2023 02 23.
Article en En | MEDLINE | ID: mdl-36780419

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Resistencia a Múltiples Medicamentos / Resistencia a Antineoplásicos / Transportador de Casetes de Unión a ATP, Subfamilia B, Miembro 2 / Proteínas de Neoplasias / Antineoplásicos Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: China

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Resistencia a Múltiples Medicamentos / Resistencia a Antineoplásicos / Transportador de Casetes de Unión a ATP, Subfamilia B, Miembro 2 / Proteínas de Neoplasias / Antineoplásicos Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: China