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A novel class of ethacrynic acid derivatives as promising drug-like potent generation of anticancer agents with established mechanism of action.
Mignani, Serge; El Brahmi, Nabil; El Kazzouli, Saïd; Eloy, Laure; Courilleau, Delphine; Caron, Joachim; Bousmina, Mosto M; Caminade, Anne-Marie; Cresteil, Thierry; Majoral, Jean-Pierre.
Afiliación
  • Mignani S; Laboratoire de Chimie et de Biochimie pharmacologiques et toxicologique, CNRS UMR 860, Université Paris Descartes, PRES Sorbonne Paris Cité, 45, rue des Saints Pères, 75006, Paris, France. Electronic address: serge.mignani@parisdescartes.fr.
  • El Brahmi N; Euromed Research Institute, Engineering Division, Euro-Mediterranean University of Fes, Fès-Shore, Route de Sidi Hrazem, 30070, Fès, Morocco; Laboratoire de Chimie de Coordination CNRS, 205 route de Narbonne, BP 44099, 31077, Toulouse Cedex 4, France; Université de Toulouse, UPS, INPT, F-31077, Toul
  • El Kazzouli S; Euromed Research Institute, Engineering Division, Euro-Mediterranean University of Fes, Fès-Shore, Route de Sidi Hrazem, 30070, Fès, Morocco. Electronic address: s.elkazzouli@ueuromed.org.
  • Eloy L; Institut de Chimie des Substances Naturelles, CNRS UPR2301, Avenue de la terrasse, 91190, Gif sur Yvette, France.
  • Courilleau D; IPSIT Faculté de Pharmacie, Université Paris Sud, 92290, Chatenay-Malabry, France.
  • Caron J; Euromed Research Institute, Engineering Division, Euro-Mediterranean University of Fes, Fès-Shore, Route de Sidi Hrazem, 30070, Fès, Morocco; Laboratoire de Chimie de Coordination CNRS, 205 route de Narbonne, BP 44099, 31077, Toulouse Cedex 4, France; Université de Toulouse, UPS, INPT, F-31077, Toul
  • Bousmina MM; Euromed Research Institute, Engineering Division, Euro-Mediterranean University of Fes, Fès-Shore, Route de Sidi Hrazem, 30070, Fès, Morocco.
  • Caminade AM; Laboratoire de Chimie de Coordination CNRS, 205 route de Narbonne, BP 44099, 31077, Toulouse Cedex 4, France; Université de Toulouse, UPS, INPT, F-31077, Toulouse Cedex4, France.
  • Cresteil T; Institut de Chimie des Substances Naturelles, CNRS UPR2301, Avenue de la terrasse, 91190, Gif sur Yvette, France; IPSIT Faculté de Pharmacie, Université Paris Sud, 92290, Chatenay-Malabry, France. Electronic address: thierry.cresteil@u-psud.fr.
  • Majoral JP; Laboratoire de Chimie de Coordination CNRS, 205 route de Narbonne, BP 44099, 31077, Toulouse Cedex 4, France; Université de Toulouse, UPS, INPT, F-31077, Toulouse Cedex4, France. Electronic address: jean-pierre.majoral@lcc-toulouse.fr.
Eur J Med Chem ; 122: 656-673, 2016 Oct 21.
Article en En | MEDLINE | ID: mdl-27448922

Texto completo: 1 Colección: 01-internacional Asunto principal: Ácido Etacrínico / Antineoplásicos Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2016 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Asunto principal: Ácido Etacrínico / Antineoplásicos Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2016 Tipo del documento: Article