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Antiviral drug screen identifies DNA-damage response inhibitor as potent blocker of SARS-CoV-2 replication.
Garcia, Gustavo; Sharma, Arun; Ramaiah, Arunachalam; Sen, Chandani; Purkayastha, Arunima; Kohn, Donald B; Parcells, Mark S; Beck, Sebastian; Kim, Heeyoung; Bakowski, Malina A; Kirkpatrick, Melanie G; Riva, Laura; Wolff, Karen C; Han, Brandon; Yuen, Constance; Ulmert, David; Purbey, Prabhat K; Scumpia, Philip; Beutler, Nathan; Rogers, Thomas F; Chatterjee, Arnab K; Gabriel, Gülsah; Bartenschlager, Ralf; Gomperts, Brigitte; Svendsen, Clive N; Betz, Ulrich A K; Damoiseaux, Robert D; Arumugaswami, Vaithilingaraja.
Afiliación
  • Garcia G; Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA 90095, USA.
  • Sharma A; Board of Governors Regenerative Medicine Institute, Cedars-Sinai Medical Center, Los Angeles, CA 90048, USA; Smidt Heart Institute, Cedars-Sinai Medical Center, Los Angeles, CA 90048, USA.
  • Ramaiah A; Department of Ecology and Evolutionary Biology, University of California, Irvine, Irvine, CA 92697, USA; Section of Cell and Developmental Biology, University of California, San Diego, San Diego, CA 92093, USA.
  • Sen C; UCLA Children's Discovery and Innovation Institute, Mattel Children's Hospital UCLA, Department of Pediatrics, David Geffen School of Medicine, UCLA, Los Angeles, CA 90095, USA.
  • Purkayastha A; UCLA Children's Discovery and Innovation Institute, Mattel Children's Hospital UCLA, Department of Pediatrics, David Geffen School of Medicine, UCLA, Los Angeles, CA 90095, USA.
  • Kohn DB; UCLA Children's Discovery and Innovation Institute, Mattel Children's Hospital UCLA, Department of Pediatrics, David Geffen School of Medicine, UCLA, Los Angeles, CA 90095, USA; Jonsson Comprehensive Cancer Center, UCLA, Los Angeles, CA 90095, USA; Eli and Edythe Broad Center of Regenerative Medicin
  • Parcells MS; Department of Animal and Food Sciences, Department of Biological Sciences, University of Delaware, Newark, DE 19716, USA.
  • Beck S; Heinrich Pette Institute, Leibniz Institute for Experimental Virology, Hamburg, Germany.
  • Kim H; Department of Infectious Diseases, Molecular Virology, Heidelberg University, Heidelberg, Germany.
  • Bakowski MA; Calibr, a division of Scripps Research Institute, 11119 North Torrey Pines Road, La Jolla, CA 92037, USA.
  • Kirkpatrick MG; Calibr, a division of Scripps Research Institute, 11119 North Torrey Pines Road, La Jolla, CA 92037, USA.
  • Riva L; Calibr, a division of Scripps Research Institute, 11119 North Torrey Pines Road, La Jolla, CA 92037, USA.
  • Wolff KC; Calibr, a division of Scripps Research Institute, 11119 North Torrey Pines Road, La Jolla, CA 92037, USA.
  • Han B; California NanoSystems Institute, University of California, Los Angeles, Los Angeles, CA 90095, USA.
  • Yuen C; California NanoSystems Institute, University of California, Los Angeles, Los Angeles, CA 90095, USA.
  • Ulmert D; Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA 90095, USA; Jonsson Comprehensive Cancer Center, UCLA, Los Angeles, CA 90095, USA.
  • Purbey PK; Department of Pathology and Laboratory Medicine, University of California, Los Angeles, Los Angeles, CA 90095, USA.
  • Scumpia P; Department of Pathology and Laboratory Medicine, University of California, Los Angeles, Los Angeles, CA 90095, USA.
  • Beutler N; Department of Immunology and Microbiology, Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, CA 92037, USA.
  • Rogers TF; Department of Immunology and Microbiology, Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, CA 92037, USA; UC San Diego Division of Infectious Diseases and Global Public Health, UC San Diego School of Medicine, La Jolla, CA 92093, USA.
  • Chatterjee AK; Calibr, a division of Scripps Research Institute, 11119 North Torrey Pines Road, La Jolla, CA 92037, USA.
  • Gabriel G; Heinrich Pette Institute, Leibniz Institute for Experimental Virology, Hamburg, Germany.
  • Bartenschlager R; Department of Infectious Diseases, Molecular Virology, Heidelberg University, Heidelberg, Germany; German Center for Infection Research, Heidelberg partner site, Heidelberg, Germany; Division Virus-Associated Carcinogenesis, German Cancer Research Center (DKFZ), Heidelberg, Germany.
  • Gomperts B; UCLA Children's Discovery and Innovation Institute, Mattel Children's Hospital UCLA, Department of Pediatrics, David Geffen School of Medicine, UCLA, Los Angeles, CA 90095, USA; Jonsson Comprehensive Cancer Center, UCLA, Los Angeles, CA 90095, USA; Eli and Edythe Broad Center of Regenerative Medicin
  • Svendsen CN; Board of Governors Regenerative Medicine Institute, Cedars-Sinai Medical Center, Los Angeles, CA 90048, USA.
  • Betz UAK; Merck KGaA, Darmstadt, Germany. Electronic address: ulrich.betz@merckgroup.com.
  • Damoiseaux RD; Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA 90095, USA; Jonsson Comprehensive Cancer Center, UCLA, Los Angeles, CA 90095, USA; California NanoSystems Institute, University of California, Los Angeles, Los Angeles, CA 90095, USA; Department
  • Arumugaswami V; Department of Molecular and Medical Pharmacology, University of California, Los Angeles, Los Angeles, CA 90095, USA; Eli and Edythe Broad Center of Regenerative Medicine and Stem Cell Research, UCLA, Los Angeles, CA 90095, USA; California NanoSystems Institute, University of California, Los Angeles,
Cell Rep ; 35(1): 108940, 2021 04 06.
Article en En | MEDLINE | ID: mdl-33784499

Texto completo: 1 Colección: 01-internacional Asunto principal: Antivirales / Pirazinas / Replicación Viral / Daño del ADN / SARS-CoV-2 / Tratamiento Farmacológico de COVID-19 / Isoxazoles Límite: Animals / Humans Idioma: En Revista: Cell Rep Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Asunto principal: Antivirales / Pirazinas / Replicación Viral / Daño del ADN / SARS-CoV-2 / Tratamiento Farmacológico de COVID-19 / Isoxazoles Límite: Animals / Humans Idioma: En Revista: Cell Rep Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos