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Identification of ARUK2002821 as an isoform-selective PI5P4Kα inhibitor.
Willems, Henriëtte M G; Edwards, Simon; Boffey, Helen K; Chawner, Stephen J; Green, Christopher; Romero, Tamara; Winpenny, David; Skidmore, John; Clarke, Jonathan H; Andrews, Stephen P.
Afiliación
  • Willems HMG; The ALBORADA Drug Discovery Institute, University of Cambridge Island Research Building, Cambridge Biomedical Campus, Hills Road Cambridge CB2 0AH UK spa26@cam.ac.uk.
  • Edwards S; The ALBORADA Drug Discovery Institute, University of Cambridge Island Research Building, Cambridge Biomedical Campus, Hills Road Cambridge CB2 0AH UK spa26@cam.ac.uk.
  • Boffey HK; The ALBORADA Drug Discovery Institute, University of Cambridge Island Research Building, Cambridge Biomedical Campus, Hills Road Cambridge CB2 0AH UK spa26@cam.ac.uk.
  • Chawner SJ; The ALBORADA Drug Discovery Institute, University of Cambridge Island Research Building, Cambridge Biomedical Campus, Hills Road Cambridge CB2 0AH UK spa26@cam.ac.uk.
  • Green C; The ALBORADA Drug Discovery Institute, University of Cambridge Island Research Building, Cambridge Biomedical Campus, Hills Road Cambridge CB2 0AH UK spa26@cam.ac.uk.
  • Romero T; The ALBORADA Drug Discovery Institute, University of Cambridge Island Research Building, Cambridge Biomedical Campus, Hills Road Cambridge CB2 0AH UK spa26@cam.ac.uk.
  • Winpenny D; The ALBORADA Drug Discovery Institute, University of Cambridge Island Research Building, Cambridge Biomedical Campus, Hills Road Cambridge CB2 0AH UK spa26@cam.ac.uk.
  • Skidmore J; The ALBORADA Drug Discovery Institute, University of Cambridge Island Research Building, Cambridge Biomedical Campus, Hills Road Cambridge CB2 0AH UK spa26@cam.ac.uk.
  • Clarke JH; The ALBORADA Drug Discovery Institute, University of Cambridge Island Research Building, Cambridge Biomedical Campus, Hills Road Cambridge CB2 0AH UK spa26@cam.ac.uk.
  • Andrews SP; The ALBORADA Drug Discovery Institute, University of Cambridge Island Research Building, Cambridge Biomedical Campus, Hills Road Cambridge CB2 0AH UK spa26@cam.ac.uk.
RSC Med Chem ; 14(5): 934-946, 2023 May 25.
Article en En | MEDLINE | ID: mdl-37252102

Texto completo: 1 Colección: 01-internacional Tipo de estudio: Diagnostic_studies Idioma: En Revista: RSC Med Chem Año: 2023 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Tipo de estudio: Diagnostic_studies Idioma: En Revista: RSC Med Chem Año: 2023 Tipo del documento: Article