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Novel N-Arylmethyl-aniline/chalcone hybrids as potential VEGFR inhibitors: synthesis, biological evaluations, and molecular dynamic simulations.
Haffez, Hesham; Elsayed, Nosaiba A; Ahmed, Marwa F; Fatahala, Samar S; Khaleel, Eman F; Badi, Rehab Mustafa; Elkaeed, Eslam B; El Hassab, Mahmoud A; Hammad, Sherif F; Eldehna, Wagdy M; Masurier, Nicolas; El-Haggar, Radwan.
Afiliación
  • Haffez H; Biochemistry and Molecular Biology Department, Faculty of Pharmacy, Helwan University, Cairo, Ain Helwan, Egypt.
  • Elsayed NA; Center of Scientific Excellence "Helwan Structural Biology Research, (HSBR)", Helwan University, Cairo, Egypt.
  • Ahmed MF; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Helwan University, Cairo, Ain Helwan, Egypt.
  • Fatahala SS; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Helwan University, Cairo, Ain Helwan, Egypt.
  • Khaleel EF; Pharmaceutical Organic Chemistry Department, Faculty of Pharmacy, Helwan University, Cairo, Egypt.
  • Badi RM; Department of Medical Physiology, College of Medicine, King Khalid University, Asir, Saudi Arabia.
  • Elkaeed EB; Department of Medical Physiology, College of Medicine, King Khalid University, Asir, Saudi Arabia.
  • El Hassab MA; Department of Pharmaceutical Sciences, College of Pharmacy, AlMaarefa University, Riyadh, Saudi Arabia.
  • Hammad SF; Department of Medicinal Chemistry, Faculty of Pharmacy, King Salman International University (KSIU), South Sinai, Egypt.
  • Eldehna WM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Helwan University, Cairo, Ain Helwan, Egypt.
  • Masurier N; Medicinal Chemistry Department, PharmD Program, Egypt-Japan University of Science and Technology (E-JUST), New Borg El-Arab City, Egypt Alexandria.
  • El-Haggar R; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, Egypt.
J Enzyme Inhib Med Chem ; 38(1): 2278022, 2023 Dec.
Article en En | MEDLINE | ID: mdl-37982203

Texto completo: 1 Colección: 01-internacional Asunto principal: Chalcona / Chalconas Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Egipto

Texto completo: 1 Colección: 01-internacional Asunto principal: Chalcona / Chalconas Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Egipto