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BPR1M97, a dual mu opioid receptor/nociceptin-orphanin FQ peptide receptor agonist, produces potent antinociceptive effects with safer properties than morphine.
Chao, Po-Kuan; Chang, Hsiao-Fu; Chang, Wan-Ting; Yeh, Teng-Kuang; Ou, Li-Chin; Chuang, Jian-Ying; Tsu-An Hsu, John; Tao, Pao-Luh; Loh, Horace H; Shih, Chuan; Ueng, Shau-Hua; Yeh, Shiu-Hwa.
Afiliação
  • Chao PK; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes, Miaoli County, 35053, Taiwan.
  • Chang HF; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes, Miaoli County, 35053, Taiwan.
  • Chang WT; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes, Miaoli County, 35053, Taiwan.
  • Yeh TK; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes, Miaoli County, 35053, Taiwan.
  • Ou LC; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes, Miaoli County, 35053, Taiwan.
  • Chuang JY; The PhD Program for Neural Regenerative Medicine, Taipei Medical University, Taipei, 110, Taiwan.
  • Tsu-An Hsu J; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes, Miaoli County, 35053, Taiwan.
  • Tao PL; Center for Neuropsychiatric Research, National Heath Research Institutes, Zhunan, Miaoli County, 35053, Taiwan.
  • Loh HH; Department of Pharmacology, University of Minnesota Medical School, Minneapolis, MN, 55455-0217, USA.
  • Shih C; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes, Miaoli County, 35053, Taiwan.
  • Ueng SH; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes, Miaoli County, 35053, Taiwan; School of Pharmacy, National Cheng Kung University, Tainan, Taiwan, ROC. Electronic address: shueng@nhri.org.tw.
  • Yeh SH; Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes, Miaoli County, 35053, Taiwan; The PhD Program for Neural Regenerative Medicine, Taipei Medical University, Taipei, 110, Taiwan. Electronic address: bau9763@nhri.org.tw.
Neuropharmacology ; 166: 107678, 2020 04.
Article em En | MEDLINE | ID: mdl-31278929

Texto completo: 1 Coleções: 01-internacional Temas: Geral Base de dados: MEDLINE Assunto principal: Medição da Dor / Receptores Opioides / Receptores Opioides mu / Analgésicos / Analgésicos Opioides / Morfina Limite: Animals / Humans / Male Idioma: En Revista: Neuropharmacology Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Taiwan

Texto completo: 1 Coleções: 01-internacional Temas: Geral Base de dados: MEDLINE Assunto principal: Medição da Dor / Receptores Opioides / Receptores Opioides mu / Analgésicos / Analgésicos Opioides / Morfina Limite: Animals / Humans / Male Idioma: En Revista: Neuropharmacology Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Taiwan