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A Fluorescent Kinase Inhibitor that Exhibits Diagnostic Changes in Emission upon Binding.
Fleming, Cassandra L; Sandoz, Patrick A; Inghardt, Tord; Önfelt, Björn; Grøtli, Morten; Andréasson, Joakim.
Afiliação
  • Fleming CL; Department of Chemistry and Chemical Engineering, Physical Chemistry, Chalmers University of Technology, 41296, Göteborg, Sweden.
  • Sandoz PA; Department of Chemistry and Molecular Biology, University of Gothenburg, 41296, Göteborg, Sweden.
  • Inghardt T; Department of Applied Physics, Science for Life Laboratory, KTH Royal Institute of Technology, 10691, Stockholm, Sweden.
  • Önfelt B; Medicinal Chemistry, Research and Early Development Cardiovascular, Renal and Metabolism, BioPharmaceuticals R&D, AstraZeneca, Gothenburg, Sweden.
  • Grøtli M; Department of Applied Physics, Science for Life Laboratory, KTH Royal Institute of Technology, 10691, Stockholm, Sweden.
  • Andréasson J; Department of Microbiology, Tumor and Cell Biology, Karolinska Institute, 17177, Stockholm, Sweden.
Angew Chem Int Ed Engl ; 58(42): 15000-15004, 2019 10 14.
Article em En | MEDLINE | ID: mdl-31411364

Texto completo: 1 Coleções: 01-internacional Temas: Geral Base de dados: MEDLINE Assunto principal: Proteína Tirosina Quinase p56(lck) Linfócito-Específica / Inibidores de Proteínas Quinases / Corantes Fluorescentes / 2-Naftilamina Tipo de estudo: Diagnostic_studies Limite: Humans Idioma: En Revista: Angew Chem Int Ed Engl Ano de publicação: 2019 Tipo de documento: Article País de afiliação: Suécia

Texto completo: 1 Coleções: 01-internacional Temas: Geral Base de dados: MEDLINE Assunto principal: Proteína Tirosina Quinase p56(lck) Linfócito-Específica / Inibidores de Proteínas Quinases / Corantes Fluorescentes / 2-Naftilamina Tipo de estudo: Diagnostic_studies Limite: Humans Idioma: En Revista: Angew Chem Int Ed Engl Ano de publicação: 2019 Tipo de documento: Article País de afiliação: Suécia