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1.
In vivo selective inhibition of TRPC6 by antagonist BI 749327 ameliorates fibrosis and dysfunction in cardiac and renal disease.
Proc Natl Acad Sci U S A
; 116(20): 10156-10161, 2019 05 14.
Article
in English
| MEDLINE | ID: mdl-31028142
2.
Mechanistic Model for the Prediction of Small-Molecule Vitreal Clearance Combining Diffusion-Limited and Permeability-Limited Clearance.
Mol Pharm
; 18(7): 2703-2713, 2021 07 05.
Article
in English
| MEDLINE | ID: mdl-34151575
3.
Carboxylesterase Activities and Protein Expression in Rabbit and Pig Ocular Tissues.
Mol Pharm
; 18(3): 1305-1316, 2021 03 01.
Article
in English
| MEDLINE | ID: mdl-33595329
4.
Quantification of Transporter and Receptor Proteins in Dog Brain Capillaries and Choroid Plexus: Relevance for the Distribution in Brain and CSF of Selected BCRP and P-gp Substrates.
Mol Pharm
; 14(10): 3436-3447, 2017 10 02.
Article
in English
| MEDLINE | ID: mdl-28880093
5.
Selective CB2 receptor agonists. Part 3: the optimization of a piperidine-based series that demonstrated efficacy in an in vivo neuropathic pain model.
Bioorg Med Chem Lett
; 25(3): 587-92, 2015 Feb 01.
Article
in English
| MEDLINE | ID: mdl-25575658
6.
Selective CB2 receptor agonists. Part 2: Structure-activity relationship studies and optimization of proline-based compounds.
Bioorg Med Chem Lett
; 25(3): 581-6, 2015 Feb 01.
Article
in English
| MEDLINE | ID: mdl-25556092
7.
LC/MS Assessment of Glycoform Clearance of A Biotherapeutic MAb in Rabbit Ocular Tissues.
J Pharm Sci
; 112(8): 2285-2291, 2023 08.
Article
in English
| MEDLINE | ID: mdl-37062414
8.
Towards holistic Compound Quality Scores: Extending ligand efficiency indices with compound pharmacokinetic characteristics.
Drug Discov Today
; 28(11): 103758, 2023 Nov.
Article
in English
| MEDLINE | ID: mdl-37660984
9.
Ocular metabolism and distribution of drugs in the rabbit eye: Quantitative assessment after intracameral and intravitreal administrations.
Int J Pharm
; 613: 121361, 2022 Feb 05.
Article
in English
| MEDLINE | ID: mdl-34896561
10.
Nanchangmycin regulates FYN, PTK2, and MAPK1/3 to control the fibrotic activity of human hepatic stellate cells.
Elife
; 112022 05 26.
Article
in English
| MEDLINE | ID: mdl-35617485
11.
1,4-Diazepane compounds as potent and selective CB2 agonists: optimization of metabolic stability.
Bioorg Med Chem Lett
; 21(7): 2011-6, 2011 Apr 01.
Article
in English
| MEDLINE | ID: mdl-21354795
12.
A Bidirectional Permeability Assay for beyond Rule of 5 Compounds.
Pharmaceutics
; 13(8)2021 Jul 27.
Article
in English
| MEDLINE | ID: mdl-34452112
13.
Quantification of Drugs in Distinctly Separated Ocular Substructures of Albino and Pigmented Rats.
Pharmaceutics
; 12(12)2020 Dec 02.
Article
in English
| MEDLINE | ID: mdl-33276439
14.
Muscle to Brain Partitioning as Measure of Transporter-Mediated Efflux at the Rat Blood-Brain Barrier and Its Implementation into Compound Optimization in Drug Discovery.
Pharmaceutics
; 11(11)2019 Nov 11.
Article
in English
| MEDLINE | ID: mdl-31718023
15.
SGLT6 - A pharmacological target for the treatment of obesity?
Adipocyte
; 7(4): 277-284, 2018.
Article
in English
| MEDLINE | ID: mdl-30161013
16.
Treatment with HC-070, a potent inhibitor of TRPC4 and TRPC5, leads to anxiolytic and antidepressant effects in mice.
PLoS One
; 13(1): e0191225, 2018.
Article
in English
| MEDLINE | ID: mdl-29385160
17.
Altered drug disposition of the platelet activating factor antagonist apafant in mdr1a knockout mice.
Eur J Pharm Sci
; 16(3): 119-28, 2002 Aug.
Article
in English
| MEDLINE | ID: mdl-12128165
18.
[The formation of a mediator of inflammation]
ALTEX
; 13(1): 17-23, 1996.
Article
in English
| MEDLINE | ID: mdl-11178441
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