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Discovery and Optimization of Orally Bioavailable Phthalazone and Cinnolone Carboxylic Acid Derivatives as S1P2 Antagonists against Fibrotic Diseases.
J Med Chem
; 64(19): 14557-14586, 2021 10 14.
Article
in English
| MEDLINE | ID: mdl-34581584
2.
Novel spirotetracyclic zwitterionic dual H(1)/5-HT(2A) receptor antagonists for the treatment of sleep disorders.
J Med Chem
; 53(21): 7778-95, 2010 Nov 11.
Article
in English
| MEDLINE | ID: mdl-20942472
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