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Bioorg Med Chem Lett
; 13(7): 1329-31, 2003 Apr 07.
Artículo
en Inglés
| MEDLINE
| ID: mdl-12657275
RESUMEN
The synthesis and antibacterial activity of benzo[f][1,7]naphtyridone derivatives are reported. These compounds are potent antibacterial agents with a Gram-positive spectrum of activity. They are active against multi-resistant cocci, especially Staphylococcus aureus strains. Their physico-chemical and biological properties make them particularly suitable for topical antibacterial use.