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1.
Novel 5-HT7 receptor antagonists modulate intestinal immune responses and reduce severity of colitis.
Am J Physiol Gastrointest Liver Physiol
; 327(1): G57-G69, 2024 Jul 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-38713616
2.
Novel druggable mechanism of Parkinson's disease: Potential therapeutics and underlying pathogenesis based on ferroptosis.
Med Res Rev
; 43(4): 872-896, 2023 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-36924451
3.
4-Oxooctahydroquinoline-1(2H)-carboxamides as hepatitis B virus (HBV) capsid core protein assembly modulators.
Bioorg Med Chem Lett
; 58: 128518, 2022 02 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-34979256
4.
MC-100093, a Novel ß-Lactam Glutamate Transporter-1 Enhancer Devoid of Antimicrobial Properties, Attenuates Cocaine Relapse in Rats.
J Pharmacol Exp Ther
; 378(2): 51-59, 2021 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-33986035
5.
Factors Governing Selectivity of Dopamine Receptor Binding Compounds for D2R and D3R Subtypes.
J Chem Inf Model
; 61(6): 2829-2843, 2021 06 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-33988991
6.
Targeting SARS-CoV-2 M3CLpro by HCV NS3/4a Inhibitors: In Silico Modeling and In Vitro Screening.
J Chem Inf Model
; 61(2): 1020-1032, 2021 02 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-33538596
7.
Design, synthesis, and evaluation of N-(4-(4-phenyl piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamides as selective dopamine D3 receptor ligands.
Bioorg Med Chem Lett
; 29(18): 2690-2694, 2019 09 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-31387791
8.
Quantum Relaxation and Metastability of Lattice Bosons with Cavity-Induced Long-Range Interactions.
Phys Rev Lett
; 121(9): 095301, 2018 Aug 31.
Artículo
en Inglés
| MEDLINE | ID: mdl-30230868
9.
Design and synthesis of functionalized piperazin-1yl-(E)-stilbenes as inhibitors of 17α-hydroxylase-C17,20-lyase (Cyp17).
Bioorg Med Chem Lett
; 28(13): 2270-2274, 2018 07 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-29803730
10.
Design, synthesis, and evaluation of (2S,4R)-Ketoconazole sulfonamide analogs as potential treatments for Metabolic Syndrome.
Bioorg Med Chem Lett
; 26(23): 5825-5829, 2016 12 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-27789139
11.
Beneficial Effect of a Small Pharmacologic Chaperone on the Established Alzheimer's Disease Phenotype.
J Alzheimers Dis
; 91(1): 463-469, 2023.
Artículo
en Inglés
| MEDLINE | ID: mdl-36442197
12.
Retromer Stabilization Improves Cognitive Function and Synaptic Plasticity in a Mouse Model of Down Syndrome.
J Alzheimers Dis
; 94(2): 513-518, 2023.
Artículo
en Inglés
| MEDLINE | ID: mdl-37334603
13.
HIV gp120 impairs nucleus accumbens neuroimmune function and dopamine D3 receptor-mediated inhibition of cocaine seeking in male rats.
Addict Neurosci
; 52023 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-36909738
14.
Riluzole prodrugs for melanoma and ALS: design, synthesis, and in vitro metabolic profiling.
Bioorg Med Chem
; 20(18): 5642-8, 2012 Sep 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-22892214
15.
Development of an amorphous based sustained release system for apremilast a selective phosphodiesterase 4 (PDE4) inhibitor.
Int J Pharm
; 615: 121516, 2022 Mar 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-35091003
16.
Antifungal properties of (2S, 4R)-Ketoconazole sulfonamide analogs.
Front Drug Discov (Lausanne)
; 22022.
Artículo
en Inglés
| MEDLINE | ID: mdl-37214226
17.
Dysfunction of the retromer complex system contributes to amyloid and tau pathology in a stem cell model of Down syndrome.
Alzheimers Dement (N Y)
; 8(1): e12334, 2022.
Artículo
en Inglés
| MEDLINE | ID: mdl-35910668
18.
Selectivity profile comparison for certain γ-butyrolactone and oxazolidinone-based ligands on a sigma 2 receptor over sigma 1: a molecular docking approach.
RSC Adv
; 12(31): 20096-20109, 2022 Jul 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-35919619
19.
5-HT1B receptor agonist enhances breakpoint for cocaine on a progressive ratio (PR) schedule during maintenance of self-administration in female rats but reduces breakpoint for sucrose.
Front Behav Neurosci
; 16: 1020146, 2022.
Artículo
en Inglés
| MEDLINE | ID: mdl-36386780
20.
Dopamine D3 receptor ligand suppresses the expression of levodopa-induced dyskinesia in nonhuman primate model of parkinson's disease.
Exp Neurol
; 347: 113920, 2022 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-34762921