1.
Bioorg Med Chem Lett
; 19(12): 3328-32, 2009 Jun 15.
Artículo
en Inglés
| MEDLINE
| ID: mdl-19442519
RESUMEN
The design and profile of a series of zwitterionic calcium sensing receptor negative allosteric modulators is described. Evaluation of key analogues using a rat model demonstrate a robust response, significantly improved potency over ronacaleret and have the potential as an oral, anabolic treatment for osteoporosis.