1.
Bioorg Med Chem Lett
; 15(15): 3501-5, 2005 Aug 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-15982875
RESUMO
A novel isoquinuclidine containing selective melanocortin subtype-4 receptor small molecule agonist, 3 (RY764), is reported. Its in vivo characterization revealed mechanism-based food intake reduction and erectile activity augmentation in rodents.