Detalhe da pesquisa
1.
Synthesis of analogs of the Gwt1 inhibitor manogepix (APX001A) and in vitro evaluation against Cryptococcus spp.
Bioorg Med Chem Lett
; 29(23): 126713, 2019 12 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-31668974
2.
A calcineurin antifungal strategy with analogs of FK506.
Bioorg Med Chem Lett
; 27(11): 2465-2471, 2017 06 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28412204
3.
Identification of biaryl sulfone derivatives as antagonists of the histamine H3 receptor: discovery of (R)-1-(2-(4'-(3-methoxypropylsulfonyl)biphenyl-4-yl)ethyl)-2-methylpyrrolidine (APD916).
Bioorg Med Chem Lett
; 22(1): 71-5, 2012 Jan 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-22172695
4.
Total synthesis of bryostatin 1.
J Am Chem Soc
; 133(4): 744-7, 2011 Feb 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-21175177
5.
A new family of H3 receptor antagonists based on the natural product Conessine.
Bioorg Med Chem Lett
; 18(4): 1490-4, 2008 Feb 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-18194865
6.
Novel H3 receptor antagonists with improved pharmacokinetic profiles.
Bioorg Med Chem Lett
; 18(14): 4133-6, 2008 Jul 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-18554904
7.
Pyran annulation: asymmetric synthesis of 2,6-disubstituted-4-methylene tetrahydropyrans.
Org Lett
; 4(7): 1189-92, 2002 Apr 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-11922815
8.
Asymmetric Total Synthesis of Rhizoxin D Financial support has been provided by the National Institutes of Health (through grant GM-28961) and by Pfizer, Inc.
Angew Chem Int Ed Engl
; 40(1): 231-234, 2001 Jan 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-11169722
9.
Asymmetric Total Synthesis of Rhizoxin D.
Angew Chem Int Ed Engl
; 40(1): 231-234, 2001 Jan 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-29711955
10.
Design and evaluation of novel biphenyl sulfonamide derivatives with potent histamine H(3) receptor inverse agonist activity.
J Med Chem
; 52(18): 5603-11, 2009 Sep 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-19722526