1.
Bioorg Med Chem Lett
; 19(15): 4022-5, 2009 Aug 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-19581086
RESUMO
A novel small molecule NPY Y2 antagonist (3) identified from high throughput screening is described. A subsequent SAR study and optimisation programme based around this molecule is also described, leading to the identification of potent and soluble pyridyl analogue 36.