Detalhe da pesquisa
1.
SAR and biological evaluation of SEN12333/WAY-317538: Novel alpha 7 nicotinic acetylcholine receptor agonist.
Bioorg Med Chem
; 17(14): 5247-58, 2009 Jul 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-19515567
2.
Base promoted isomerization of aziridinyl ethers: a new access to alpha- and beta-amino acids.
Chem Commun (Camb)
; (7): 778-9, 2002 Apr 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-12119719
3.
Fused 3-Hydroxy-3-trifluoromethylpyrazoles Inhibit Mutant Huntingtin Toxicity.
ACS Med Chem Lett
; 4(10): 979-84, 2013 Oct 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-24900595
4.
N-[5-(5-fluoropyridin-3-yl)-1H-pyrazol-3-yl]-4-piperidin-1-ylbutyramide (SEN78702, WYE-308775): a medicinal chemistry effort toward an α7 nicotinic acetylcholine receptor agonist preclinical candidate.
J Med Chem
; 55(22): 10277-81, 2012 Nov 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-23083093
5.
Discovery of a novel alpha-7 nicotinic acetylcholine receptor agonist series and characterization of the potent, selective, and orally efficacious agonist 5-(4-acetyl[1,4]diazepan-1-yl)pentanoic acid [5-(4-methoxyphenyl)-1H-pyrazol-3-yl] amide (SEN15924, WAY-361789).
J Med Chem
; 55(10): 4806-23, 2012 May 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-22468936
6.
Novel alpha-7 nicotinic acetylcholine receptor agonists containing a urea moiety: identification and characterization of the potent, selective, and orally efficacious agonist 1-[6-(4-fluorophenyl)pyridin-3-yl]-3-(4-piperidin-1-ylbutyl) urea (SEN34625/WYE-103914).
J Med Chem
; 53(11): 4379-89, 2010 Jun 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-20465311
7.
A Selective Access to Amino Hydroxy Oxetanes.
J Org Chem
; 62(24): 8557-8559, 1997 Nov 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-11672003