Detalhe da pesquisa
1.
Rh(III)-Catalyzed C7-Alkylation of Isatogens with Malonic Acid Diazoesters.
J Org Chem
; 89(5): 2984-2995, 2024 Mar 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-38334453
2.
The Discovery of Indole-2-carboxylic Acid Derivatives as Novel HIV-1 Integrase Strand Transfer Inhibitors.
Molecules
; 28(24)2023 Dec 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-38138510
3.
Synthesis and antibiofilm evaluation of N-acyl-2-aminopyrimidine derivatives against Acinetobacter baumannii.
Bioorg Med Chem
; 76: 117095, 2022 12 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-36442439
4.
Design, Synthesis, and Biological Evaluation of N14-Amino Acid-Substituted Tetrandrine Derivatives as Potential Antitumor Agents against Human Colorectal Cancer.
Molecules
; 27(13)2022 Jun 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-35807286
5.
Discovery of tetrandrine derivatives as tumor migration, invasion and angiogenesis inhibitors.
Bioorg Chem
; 101: 104025, 2020 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-32599368
6.
Organocatalytic Asymmetric α-Sulfenylation of 2-Substituted Indolin-3-ones: A Strategy for the Synthesis of Chiral 2,2-Disubstituted Indole-3-ones with S- and N-Containing Heteroquaternary Carbon Stereocenter.
J Org Chem
; 84(12): 8168-8176, 2019 06 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-31192597
7.
Design, synthesis, and biological evaluation of 2-amino-N-(2-methoxyphenyl)-6-((4-nitrophenyl)sulfonyl)benzamide derivatives as potent HIV-1 Vif inhibitors.
Bioorg Med Chem Lett
; 29(24): 126638, 2019 12 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-31685340
8.
Design, synthesis, and cytotoxic activity of novel 7-substituted camptothecin derivatives incorporating piperazinyl-sulfonylamidine moieties.
Bioorg Med Chem Lett
; 27(17): 3959-3962, 2017 09 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28789891
9.
Design, synthesis and biological evaluation of indole-2-carboxylic acid derivatives as novel HIV-1 integrase strand transfer inhibitors.
RSC Adv
; 14(13): 9020-9031, 2024 Mar 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-38500630
10.
Synthesis of diarylmethyl thioethers via a DABCO-catalyzed 1,6-conjugate addition reaction of p-quinone methides with organosulfur reagents.
RSC Adv
; 13(19): 12982-12990, 2023 Apr 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-37124019
11.
Facilitated Drug Repurposing with Artemisinin-Derived PROTACs: Unveiling PCLAF as a Therapeutic Target.
J Med Chem
; 66(16): 11335-11350, 2023 08 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-37552639
12.
A solid-supported organocatalyst for asymmetric Mannich reaction to construct C2-quaternary indolin-3-ones.
RSC Adv
; 12(12): 7040-7045, 2022 Mar 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-35424681
13.
Synthesis and antibacterial activity studies in vitro of indirubin-3'-monoximes.
RSC Adv
; 12(38): 25068-25080, 2022 Aug 30.
Artigo
em Inglês
| MEDLINE | ID: mdl-36199871
14.
Discovery of ß-Carboline Derivatives as a Highly Potent Cardioprotectant against Myocardial Ischemia-Reperfusion Injury.
J Med Chem
; 64(13): 9166-9181, 2021 07 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-34132541
15.
Design, synthesis, and biological evaluation of 2,4-diamino pyrimidine derivatives as potent FAK inhibitors with anti-cancer and anti-angiogenesis activities.
Eur J Med Chem
; 222: 113573, 2021 Oct 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-34091209
16.
Enantioselective amination of 4-alkylisoquinoline-1,3(2H,4H)-dione derivatives.
RSC Adv
; 10(70): 42912-42915, 2020 Nov 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-35514906
17.
Catalyst-free Cleavage of Amide and C-O Double Bond for the Diastereoselective Synthesis of Trifluoromethyl-Containing Dihydrooxazole Derivatives.
Org Lett
; 21(7): 2236-2240, 2019 04 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-30859824
18.
Palladium-catalyzed direct C(sp3)-H arylation of indole-3-ones with aryl halides: a novel and efficient method for the synthesis of nucleophilic 2-monoarylated indole-3-ones.
RSC Adv
; 8(45): 25292-25297, 2018 Jul 16.
Artigo
em Inglês
| MEDLINE | ID: mdl-35539771
19.
Design, synthesis, cytotoxic activity and molecular docking studies of new 20(S)-sulfonylamidine camptothecin derivatives.
Eur J Med Chem
; 115: 109-20, 2016 Jun 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-26994847
20.
Asymmetric organocatalytic relay cascades: catalyst-controlled stereoisomer selection in the synthesis of functionalized cyclohexanes.
Angew Chem Int Ed Engl
; 48(52): 9834-8, 2009.
Artigo
em Inglês
| MEDLINE | ID: mdl-19946924