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Structure-activity studies in the development of a hydrazone based inhibitor of adipose-triglyceride lipase (ATGL).
Mayer, Nicole; Schweiger, Martina; Melcher, Michaela-Christina; Fledelius, Christian; Zechner, Rudolf; Zimmermann, Robert; Breinbauer, Rolf.
Affiliation
  • Mayer N; Institute of Organic Chemistry, Graz University of Technology, Stremayrgasse 9, A-8010 Graz, Austria.
  • Schweiger M; Institute of Molecular Biosciences, University of Graz, Heinrichstraße 31/II, A-8010 Graz, Austria.
  • Melcher MC; Institute of Organic Chemistry, Graz University of Technology, Stremayrgasse 9, A-8010 Graz, Austria.
  • Fledelius C; Novo Nordisk A/S, Novo Nordisk Park, DK-2760 Måløv, Denmark.
  • Zechner R; Institute of Molecular Biosciences, University of Graz, Heinrichstraße 31/II, A-8010 Graz, Austria.
  • Zimmermann R; Institute of Molecular Biosciences, University of Graz, Heinrichstraße 31/II, A-8010 Graz, Austria. Electronic address: robert.zimmermann@uni-graz.at.
  • Breinbauer R; Institute of Organic Chemistry, Graz University of Technology, Stremayrgasse 9, A-8010 Graz, Austria. Electronic address: breinbauer@tugraz.at.
Bioorg Med Chem ; 23(12): 2904-16, 2015 Jun 15.
Article in En | MEDLINE | ID: mdl-25778769

Full text: 1 Database: MEDLINE Main subject: Enzyme Inhibitors / Hydrazones / Lipase Limits: Animals Language: En Journal: Bioorg Med Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2015 Type: Article Affiliation country: Austria

Full text: 1 Database: MEDLINE Main subject: Enzyme Inhibitors / Hydrazones / Lipase Limits: Animals Language: En Journal: Bioorg Med Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2015 Type: Article Affiliation country: Austria