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Precise prediction of activators for the human constitutive androstane receptor using structure-based three-dimensional quantitative structure-activity relationship methods.
Kato, Harutoshi; Yamaotsu, Noriyuki; Iwazaki, Norihiko; Okamura, Shigeaki; Kume, Toshiyuki; Hirono, Shuichi.
Affiliation
  • Kato H; School of Pharmacy, Kitasato University, Minato-ku, Tokyo 108-8641, Japan; DMPK Research Laboratories, Mitsubishi Tanabe Pharma Corporation, Toda-shi, Saitama 335-8505, Japan. Electronic address: Kato.Harutoshi@mb.mt-pharma.co.jp.
  • Yamaotsu N; School of Pharmacy, Kitasato University, Minato-ku, Tokyo 108-8641, Japan.
  • Iwazaki N; DMPK Research Laboratories, Mitsubishi Tanabe Pharma Corporation, Toda-shi, Saitama 335-8505, Japan.
  • Okamura S; DMPK Research Laboratories, Mitsubishi Tanabe Pharma Corporation, Toda-shi, Saitama 335-8505, Japan.
  • Kume T; Discovery Technology Laboratories, Mitsubishi Tanabe Pharma Corporation, Toda-shi, Saitama 335-8505, Japan.
  • Hirono S; School of Pharmacy, Kitasato University, Minato-ku, Tokyo 108-8641, Japan. Electronic address: hironos@pharm.kitasato-u.ac.jp.
Drug Metab Pharmacokinet ; 32(3): 179-188, 2017 Jun.
Article in En | MEDLINE | ID: mdl-28412023

Full text: 1 Database: MEDLINE Main subject: Receptors, Cytoplasmic and Nuclear / Quantitative Structure-Activity Relationship Type of study: Prognostic_studies / Risk_factors_studies Limits: Humans Language: En Journal: Drug Metab Pharmacokinet Journal subject: FARMACOLOGIA / METABOLISMO Year: 2017 Type: Article

Full text: 1 Database: MEDLINE Main subject: Receptors, Cytoplasmic and Nuclear / Quantitative Structure-Activity Relationship Type of study: Prognostic_studies / Risk_factors_studies Limits: Humans Language: En Journal: Drug Metab Pharmacokinet Journal subject: FARMACOLOGIA / METABOLISMO Year: 2017 Type: Article